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2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylacetamide
5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylic acid
N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
1-[(2-methoxyphenyl)methyl]-N3-(3-methoxypropyl)-N5-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
5-methyl-N-(pyridin-2-ylmethyl)-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
2-(4-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-(3-methylbut-2-en-1-yl)piperazin-2-yl)ethan-1-ol
2,3-dimethyl-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-indole-7-carboxamide
(3S,4R)-1-(2,1,3-benzoxadiazol-4-ylmethyl)-4-(pyridin-3-yl)pyrrolidine-3-carboxylic acid
(2S,4R)-4-amino-N-methyl-1-[(5-propylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
(E)-N-[(7S,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2-phenylethene-1-sulfonamide
7-[2-(3-ethoxyphenoxy)ethyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
4-fluoro-N-[1-(5-{[2-(4-fluorophenoxy)ethyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]benzamide
methyl 8-[(6-chloro-4-oxo-4H-chromen-3-yl)methyl]-1-ethoxy-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
3-[(3-chlorophenyl)methyl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine-3-carboxylic acid
6-[3-(furan-2-yl)propanoyl]-N-[4-(1H-pyrazol-1-yl)phenyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(ethylsulfanyl)-1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}propan-1-one
2-{[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-5-methoxy-4H-pyran-4-one
5,6-dimethyl-3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydropyridin-2-one
N-(1,3-dihydroxypropan-2-yl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
N,N-dimethyl-4-{2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-amine
2-(methoxymethyl)-5-[(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)methyl]pyrimidine
(1S,5R)-6-{imidazo[1,2-a]pyridine-6-carbonyl}-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
4-(1H-indol-2-ylmethyl)-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-(1H-imidazol-4-ylmethyl)-2-(3-methoxypropyl)piperidine
N-[(6-methylpyridin-2-yl)methyl]-1-(piperidin-1-yl)cyclohexane-1-carboxamide
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
N-(1-phenylbutyl)-3-(5-{[3-(trifluoromethyl)phenyl]methyl}-1,3,4-oxadiazol-2-yl)propanamide
N-[4-(methylsulfanyl)phenyl]-4-(2-phenoxyacetyl)piperazine-1-carboxamide
N-ethyl-2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methylacetamide
N-(1-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperidin-4-yl)methanesulfonamide
[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl](thiophen-2-yl)methanol
4-chloro-2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]methyl}phenol
1-(4-chlorophenyl)-N-cyclopropyl-N-{[7-fluoro-2-(morpholin-4-yl)quinolin-3-yl]methyl}cyclopropane-1-carboxamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
N-[(3R,5S)-1-benzyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
methyl 4-[2-(dimethylamino)-2-(4-fluorophenyl)acetyl]piperazine-1-carboxylate
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2,6,8-trimethylquinoline-4-carboxamide
2-[(4aS,8aR)-1-(3-methylbutyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
1-cyclopropyl-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
3-[(3S,4R)-1-[(3-chlorophenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]-1-[4-(2-methoxyphenyl)piperazin-1-yl]propan-1-one
5-(1-methoxypropyl)-3-(5-methylfuran-2-yl)-1-propyl-1H-1,2,4-triazole
N-{3-[2-methoxy-5-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-acetamidopropanamide
4-[(4-fluorophenyl)methyl]-1-(6-methylpyridine-2-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
N-cyclopropyl-1-[1-(pyrimidine-5-carbonyl)piperidin-4-yl]-1H-1,2,3-triazole-4-carboxamide
1-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3-methoxy-1,2-dihydropyridin-2-one
3-{1-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(3-fluorophenyl)urea
(4aR,6R,8aS)-8a-(methoxymethyl)-2-[(1-methyl-1H-pyrazol-4-yl)methyl]-6-(morpholin-4-yl)-decahydroisoquinoline