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2-{3-[(dimethylamino)methyl]-3-hydroxypiperidine-1-carbonyl}pyridin-3-ol
N-(1-{2-[4-(3-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-(phenylsulfanyl)acetamide
4-{[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-3-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
N-[(2,6-dimethylpyridin-4-yl)methyl]-4-(piperidin-1-yl)butanamide
1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
2-amino-1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-2-methylpropan-1-one
(1-{2-[2-(1H-1,3-benzodiazol-2-yl)-1H-imidazol-1-yl]ethyl}piperidin-2-yl)methanol
1-{3,9-diazaspiro[5.5]undecan-3-yl}-3-(piperazin-1-yl)propan-1-one
(3S,4S)-1-[(5-cyano-1-ethyl-1H-pyrrol-3-yl)methyl]-4-propylpyrrolidine-3-carboxylic acid
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
N-(1-hydroxy-2-methylpropan-2-yl)-5-[3-(trifluoromethyl)phenoxymethyl]-1,2-oxazole-3-carboxamide
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-(2,5-difluorophenyl)-5-[(2-methoxyethyl)sulfamoyl]benzoic acid
1-[4-({4-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)piperazin-1-yl]ethan-1-one
2-{5-[1-(3-methoxy-2-methylbenzoyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
5-{2-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
6-{[3-(benzyloxy)phenyl]methyl}-N-(2-phenylethyl)-6-azaspiro[2.5]octane-1-carboxamide
N-[2-(4-chlorophenyl)-2-(piperidin-1-yl)ethyl]-4-methylpyrimidine-5-carboxamide
dimethyl(1-{4-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenyl}ethyl)amine
4-methyl-3-(3,4,5-trimethoxyphenyl)-1,2-dihydroquinolin-2-one
5-[4-(3-hydroxypyrrolidin-1-yl)pyrimidin-2-yl]thiophene-2-carboxylic acid
3-{[3-(methanesulfonylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,4,7-trimethyl-1H-indole
3-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}propanamide
methyl 3-[(3S,4R)-1-[(4-methylphenyl)methyl]-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]propanoate
2-(pyridin-3-yl)-N-(pyridin-3-ylmethyl)-5,6,7,8-tetrahydroquinazolin-5-amine
4-{4-[(4-chloro-3-fluorophenyl)methyl]piperazin-1-yl}butan-1-ol
N-[(2R,3R)-1'-[(3,5-dimethoxyphenyl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
8-(5-methylhex-5-en-2-yl)-1-(2-methylpropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-(4-chlorophenyl)-1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-4-ol
2-[5-(4-fluorophenyl)-1H-indol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
5-ethyl-3-[2-(4-methoxyphenyl)ethyl]-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
3-phenyl-1-{3-[(quinoxalin-2-yl)amino]azepan-1-yl}propan-1-one
N-ethyl-2,5-dimethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
3-[(dimethylamino)methyl]-1-(1H-indol-5-ylmethyl)pyrrolidin-3-ol
1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-5-oxopyrrolidine-3-carboxylic acid
N-(cyclopropylmethyl)-5-methyl-N-propyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-({3-[4-(morpholin-4-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
N-[(3S,4S)-1-ethyl-4-methoxypyrrolidin-3-yl]-3,5,7-trimethyl-1H-indole-2-carboxamide
N-butyl-N-methyl-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}cyclopropanamine
methyl 2-[2-(2-methylpropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]pyridine-3-carboxylate
2-{3-methyl-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl}benzene-1,3-diol
3-methyl-8-(2,4,5-trifluorobenzenesulfonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-1-(2-methoxyethyl)-5-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
ethyl({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
2-{1-[(5-ethylpyridin-2-yl)methyl]pyrrolidin-3-yl}benzoic acid
5-(2-methylphenyl)-2-(pyridin-3-yl)-4-[1-(1,3-thiazole-5-carbonyl)piperidin-4-yl]pyrimidine