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2-{1-[(5-methylfuran-2-yl)methyl]-4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl}ethan-1-ol
N-methyl-3-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}pyridin-2-amine
6-methoxy-N-[2-(pyridin-3-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]hexanamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-2-ylmethyl)amine
2,4-dimethoxy-6-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}pyrimidine
{4-[(4-fluoro-3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methanol
2-amino-3-ethyl-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[(4-methoxypyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
4-(1,3-dimethyl-1H-pyrazol-5-yl)-3-(oxan-4-yl)-4H-1,2,4-triazole
3-{2-[3-(4-chlorophenyl)piperidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
8-(1-benzothiophen-2-ylmethyl)-1-[2-(4-methoxyphenyl)ethyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-[(1-methyl-1,2,5,6-tetrahydropyridin-3-yl)methyl]piperidine-1-carboxamide
N-(1H-1,3-benzodiazol-2-yl)-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]acetamide
1-methyl-4-{[6-(3-methyl-3-phenylpiperidin-1-yl)pyridin-3-yl]methyl}piperazine
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-[(4-phenylphenyl)methyl]acetamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
2-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenol
methyl 9-(oxan-2-ylmethoxy)-7-oxo-3-{[4-(pyrrolidin-1-yl)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-amino-3-{2-[(oxolan-2-ylmethyl)amino]pyrimidin-5-yl}-1,6-diazatricyclo[6.2.2.02,7]dodeca-2,4,6-triene-4-carbonitrile
[4-(2-phenoxyethyl)-1-(quinolin-8-ylmethyl)piperidin-4-yl]methanol
(2S,4R)-1-[(4-fluorophenyl)methyl]-4-[(4-fluorophenyl)sulfanyl]-N,N-dimethylpyrrolidine-2-carboxamide
N-(4-{1-[2-(N-methylmethanesulfonamido)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
N-cyclopropyl-2-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)oxy]-4-methoxybenzamide
1-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-(hydroxymethyl)piperidin-3-ol
N-(adamantan-1-ylmethyl)-1-ethyl-N-methyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[3-(1H-imidazol-2-yl)benzoyl]-1-(4-methylphenyl)piperazin-2-one
N-[(3S,4R)-4-(5-methylfuran-2-yl)-1-{[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}pyrrolidin-3-yl]acetamide
(2R,3R,6R)-3-(4-fluorophenyl)-5-(4-methyl-1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[4-({4-[(3-fluorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)phenyl]acetamide
4-(4-aminopyrimidin-2-yl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
1-(cyclohexylmethyl)-6-oxo-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-3-carboxamide
ethyl 1-(5-methyl-1H-indazole-3-carbonyl)-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
9-methoxy-3-(naphthalen-1-ylmethyl)-10-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
N-[(4-fluorophenyl)methyl]-1-methyl-5-{[2-(pyridin-4-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(3aS,7aR)-2-[5-(methoxymethyl)furan-2-carbonyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-({[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]carbamoyl}amino)-N,N,3-trimethylbenzamide
N-methyl-N-[(3-methylthiophen-2-yl)methyl]-1H-indazole-3-carboxamide
1-[(3-fluoro-4-methoxyphenyl)methyl]-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
(3S,4R)-4-methyl-1-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]piperidine-3,4-diol
2-methoxy-1-{1'-[(2S)-1-methylpyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-3-yl}methyl)cycloheptanecarboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1-(2-phenylethyl)-1H-1,2,3-triazole-4-carboxamide
6-[2-(dimethylamino)phenyl]-N,N-dimethylpyridine-3-carboxamide
(3aR,6aR)-2-[2-(3-methyl-2-oxo-1,2,3,4-tetrahydroquinazolin-1-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(methoxymethyl)-1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidine
3-amino-N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-1H-1,2,4-triazole-5-carboxamide
6-ethyl-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-2-methylquinoline
1-(pyridin-3-ylmethyl)-4-[5-(trifluoromethyl)pyridin-2-yl]piperazine
N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide