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N-[(3-methyloxetan-3-yl)methyl]-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
5-(methoxymethyl)-N-{4-[5-methyl-4-({[(1R,2R)-2-phenylcyclopropyl]formamido}methyl)-1,3-oxazol-2-yl]phenyl}furan-2-carboxamide
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(2-methoxyphenyl)ethyl]acetamide
2-[3-(1H-pyrazol-3-yl)phenyl]quinoxaline
2-{[4-(ethoxymethyl)piperidin-1-yl]sulfonyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
methyl[3-(1H-pyrazol-1-yl)propyl][2-(pyridin-4-yl)ethyl]amine
6-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-oxo-2-(2-phenylethyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
3-[(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]pyridine
N-[2-(methylsulfanyl)phenyl]-3-(2-phenylacetyl)piperidine-1-carboxamide
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-8-fluoroquinoline-2-carboxamide
2-(4-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}phenyl)pyridine
[(3R,4R)-4-[(dimethylamino)methyl]-1-[4-(propan-2-yloxy)benzoyl]pyrrolidin-3-yl]methanol
(2R)-2-{4-phenyl-5-[5-(1H-pyrazol-5-yl)furan-2-yl]-1H-imidazol-1-yl}propanamide
9-[2-(1H-pyrazol-1-yl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
5-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-5-[(3-methoxyphenyl)methyl]-3-methylimidazolidine-2,4-dione
4-methyl-1-[(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-1,2,3,6-tetrahydropyridine
N-(cyclopropylmethyl)-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-propylpropanamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(6-methylpyridine-2-carbonyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(1-benzyl-1H-imidazol-2-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
7-(2,6-dimethoxyphenyl)-9-methoxy-4-(pyridin-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{2-[2-amino-3-cyano-6-(propan-2-yl)pyridin-4-yl]-4-chlorophenoxy}acetamide
(3aR,5R,6S,7aS)-2-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-isoindole-5,6-diol
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
1-(4-{[4-(4-ethylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenyl)ethan-1-one
5-(3-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
(4aS,7aR)-1-[(7-hydroxyquinolin-3-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aS,8aR)-6-[(2-aminopyrimidin-5-yl)methyl]-1-[2-(1H-imidazol-4-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
3-(4-chloro-2-methylbenzoyl)-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidine
1-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]azonan-2-one
5-phenyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-[3-(1H-indazol-1-yl)propyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-cyclobutyl-3-[3-(propan-2-yloxy)benzoyl]piperidine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[(5-fluoro-2-methylphenyl)methyl]piperidine-3-carboxamide
N-(furan-2-ylmethyl)-4-methyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}benzamide
1-pentanoyl-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{2-[(pyridin-3-yl)amino]ethyl}-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
(1-{[4-(azepan-1-yl)quinazolin-2-yl]methyl}piperidin-4-yl)methanol
({6-chloro-2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]imidazo[1,2-a]pyridin-3-yl}methyl)(methyl)(thiophen-2-ylmethyl)amine
{1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(3-phenylpropyl)piperidin-3-yl}methanol
3-[1-(naphthalene-2-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
(1S,5R)-6-(cyclopropylmethyl)-3-{2-[4-(methylsulfanyl)phenyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[(3R,4S)-4-(dimethylamino)-1-[(2-phenylethyl)carbamoyl]piperidin-3-yl]propanoic acid
1-[(3-methoxyphenyl)methyl]-4-(1H-pyrrole-3-carbonyl)piperazin-2-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-(propan-2-yl)acetamide
N-{2-[1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidin-2-yl]ethyl}acetamide
1-[2-(dimethylamino)ethyl]-5-oxo-N-(1-phenylpiperidin-4-yl)pyrrolidine-3-carboxamide
N-[(2-benzyl-1,3-thiazol-4-yl)methyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-(1,2-oxazole-3-carbonyl)-8-azabicyclo[3.2.1]octane
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-pyrrole-2-carbonyl)piperidine
(3R,4S)-1-(5-fluoro-2-methoxybenzoyl)-4-propylpyrrolidin-3-amine