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5-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
(4aR,7aS)-1-benzyl-4-[2-(pyridin-3-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2-chlorophenyl)-1-(3-methoxypropyl)-3-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}pyrrolidine-2,5-dione
2-(dimethylamino)-N-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]-2,3-dihydro-1H-indene-2-carboxamide
N-(3-{2-[(4-fluorophenyl)methyl]morpholine-4-carbonyl}phenyl)acetamide
3-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidin-3-yl)-1-(4-methylpiperazin-1-yl)propan-1-one
4-chloro-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-2-(pyrrolidin-1-yl)-1,3-thiazole
N-(1-{7-[(2-hydroxy-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)-3,5-dimethylbenzamide
1-[4-(furan-2-yl)butan-2-yl]-4-phenyl-5-(trimethyl-1H-pyrazol-4-yl)-1H-imidazole
(5S,9aS,9bS)-5-(4-fluoro-3-methoxyphenyl)-2-methyl-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-(3-methylbutyl)-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(3-ethyl-1,2-oxazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(4-{[2-(2-fluorophenyl)-1H-imidazol-1-yl]methyl}phenyl)methanamine
(4aR,8aR)-2-cyclopentanecarbonyl-7-[5-fluoro-2-(hydroxymethyl)pyridin-4-yl]-decahydro-2,7-naphthyridin-4a-ol
5-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methylphenol
{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}piperidine-4-carboxamide
1-(1-benzylpyrrolidin-3-yl)-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
N-benzyl-N-methyl-1-{[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carbonyl}piperidine-4-carboxamide
N-[2-(furan-2-yl)ethyl]-7-(2-methoxyacetamido)-1-(2-phenylethyl)-1H-1,3-benzodiazole-5-carboxamide
{[4-(1H-imidazol-1-yl)phenyl]methyl}(methyl)[2-(morpholin-4-yl)propyl]amine
8-[(4-fluorophenyl)methyl]-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-fluorophenyl)ethan-1-one
1-(1-cycloheptylpiperidin-3-yl)-3-ethylurea
N-({1-[(3-chloropyridin-4-yl)methyl]piperidin-3-yl}methyl)-1H-pyrrole-2-carboxamide
2-(piperidine-1-carbonyl)-6-(pyridin-4-yl)pyrazine
2-[2-(1-{[2-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[(2,5-dimethoxyphenyl)methyl]acetamide
N,N-dimethyl-6-[2-(pyridin-2-yl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-{2-[(5-ethyl-2-methylpyrimidin-4-yl)amino]ethyl}-1,3-oxazinan-2-one
7-methoxy-3-{[3-(2-methylpropyl)morpholin-4-yl]methyl}-1,2-dihydroquinolin-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-4-(naphthalen-2-ylmethyl)-1,4-diazepan-5-one
N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
2-cyclopropyl-8-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-5-methylphenol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-methyl-5-sulfamoylbenzamide
4-{2-[(4aR,7aS)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-2-oxoethoxy}benzoic acid
2-{1-[4-(1H-pyrazol-3-yl)benzoyl]pyrrolidin-2-yl}-1,3-thiazole
N-[2-(4-fluorophenyl)-1-[1-(quinoxaline-6-carbonyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
1-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(6-methoxy-2H-1,3-benzodioxol-5-yl)urea
2-(methylsulfanyl)-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
4-(2,5-difluorophenyl)-3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(5S,9aS,9bS)-5-(2-methoxyphenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[3-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)propyl]piperidin-3-ol
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-[(3-phenyl-1H-pyrazol-5-yl)methyl]acetamide
2-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyridine-3-carboxamide
1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-amino-7-(8-chloroquinoline-2-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
[(2S,6S)-4-(2-ethoxypyridine-3-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
2-[2,5-dioxo-3-phenyl-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)acetamide