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1-ethyl-5-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]piperidin-2-one
[(4-methoxyphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
3-methoxy-1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(2-methoxyethyl)-1-methyl-5-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1H-1,3-benzodiazol-2-amine
4-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-5-(propan-2-yl)pyrimidine
N,1-dimethyl-N-(1-{1-[(2-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-3-carboxamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]propanamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(thiophen-3-ylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-4-amino-1-(3-{[(4-fluorophenyl)methyl]sulfanyl}propanoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-methyl-6-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-5-(prop-2-en-1-yl)pyrimidin-2-amine
{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]methylamine
{9-[(5-methylthiophen-2-yl)methyl]-3-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
3-[(2-chloro-6-fluorophenyl)methyl]-9-methoxy-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-5-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]propan-2-ol
4-[1-(methoxymethyl)cyclobutaneamido]-N-phenylpiperidine-1-carboxamide
({4-ethyl-5-[1-(1H-indol-5-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
1-[1-(2-fluorobenzoyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
1-[4-(2-methylpropyl)benzoyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
5-[cyclopropyl({5-[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]-4-phenyl-1H-imidazol-1-yl})methyl]-1-methyl-1H-1,2,4-triazole
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-2-propyl-1,3-thiazole-4-carboxamide
{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}(methyl)(thiophen-3-ylmethyl)amine
1-(3-fluoro-5-methylphenyl)-3-[2-(1-hydroxycyclopentyl)ethyl]-3-methylurea
1-[(1-{[(1s,4s)-4-aminocyclohexyl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
6-ethoxy-3-{[4-(pyridin-4-yl)piperazin-1-yl]methyl}-1,2-dihydroquinolin-2-one
N-cyclopropyl-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-4-yl}propanamide
N-methyl-4-(pyrrolidine-1-carbonyl)-6-(thiophene-3-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
5-fluoro-4-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]quinazoline
2-amino-N-{2-fluoro-4-[4-(1-methoxyethyl)phenyl]phenyl}acetamide
1-[7-(3-chloro-1,2-oxazole-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]-1,2,3,6-tetrahydropyridine
[(1,5-dimethyl-1H-pyrazol-4-yl)methyl][(3-ethenylphenyl)methyl]methylamine
2-(methylamino)-1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-(pyridin-3-yl)ethan-1-one
N-cyclopropyl-3-[5-(1-phenylcyclopropanecarbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(2-methyl-1H-imidazol-1-yl)acetamide
4-{3-[(3R,4S)-3-acetamido-4-propylpyrrolidin-1-yl]propoxy}benzamide
1-{2-[3-(6-methoxynaphthalene-2-carbonyl)piperidin-1-yl]ethyl}pyrrolidin-2-one
4-(9H-fluoren-2-ylmethyl)-9-methoxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[4-({[(2,4-difluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
3-[(ethylamino)methyl]-1-{[3-(trifluoromethyl)phenyl]methyl}-1H,2H,6H,7H,8H-cyclopenta[g]quinolin-2-one
(4aS,7aR)-1-[2-(3-hydroxyphenyl)acetyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]piperidine-1-carbonyl}pyridine
8-(dimethyl-1,3-thiazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
2,5,7-trimethyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}quinoline-4-carboxamide
methyl({1-[(1-pentylpiperidin-3-yl)methyl]-1H-1,2,3-triazol-4-yl}methyl)amine
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-methyl-8-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2,3-dimethoxyphenyl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine