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2-(dimethylamino)-8-(4-fluoro-3-methylphenyl)-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-ethyl-N-[3-(furan-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(thiophene-3-carbonyl)piperidin-3-ol
2-{3-cyclopropyl-5-[2-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}-4-methylpyridine
1-methyl-5-[methyl(thiophen-3-ylmethyl)amino]-N-[2-(morpholin-4-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-cyclopropyl-4-phenyl-9-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)benzamide
N,N,4-trimethyl-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
2-(2-hydroxyethyl)-9-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(1,2-benzoxazol-3-yl)-N-[2-(pyridin-3-yloxy)ethyl]acetamide
2-(4-chlorophenyl)-1-[3-(morpholine-4-carbonyl)-1-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]ethan-1-one
3-(5-fluoro-2-methoxybenzoyl)-1-(4-methyl-1,3-oxazole-5-carbonyl)piperidine
1-{7-[cyclohexyl(hydroxy)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-(phenylsulfanyl)ethan-1-one
N-[(2R,3R)-1'-(4-acetylbenzoyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-5-methyl-5-{1-[(3-methylthiophen-2-yl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
N-(1-phenylbutyl)azetidine-3-carboxamide
(3S,5R)-N3-butyl-N5-(4-fluorophenyl)-1-[(4-hydroxyphenyl)methyl]piperidine-3,5-dicarboxamide
2-(5-acetylthiophen-3-yl)-1-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]ethan-1-one
2-{4-[(4-chlorophenyl)methyl]-1-(3-methylbut-2-en-1-yl)piperazin-2-yl}ethan-1-ol
3-butyl-1-methyl-4-({7-methylimidazo[1,2-a]pyridin-2-yl}methyl)piperazin-2-one
N-[(1-ethylpiperidin-2-yl)methyl]-5,6-dimethylpyrimidin-4-amine
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(propan-2-yl)pyrimidine-5-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-2-propyl-1,3-thiazole-4-carboxamide
{[5-(1-cyclooctylpiperidin-4-yl)-4-cyclopropyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine
3-(2-chlorophenyl)-5-methyl-N-[(6-oxo-1,6-dihydropyrimidin-4-yl)methyl]-1,2-oxazole-4-carboxamide
7-fluoro-3-(1-methyl-2-oxopyrrolidin-3-yl)-3,4-dihydroquinazolin-4-one
ethyl 1-(3-phenylpropyl)-5-(1H-pyrazol-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-chloro-N-[1-(pyrimidin-2-yl)piperidin-3-yl]pyridine-4-carboxamide
3-[3-(furan-3-yl)phenyl]-1-[(1-methyl-1H-imidazol-5-yl)methyl]-1H-pyrazole
2-{4-methyl-2-[3-(pyridin-3-yl)-1H-pyrazol-1-yl]phenoxy}acetamide
N-(butan-2-yl)-1-ethyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]amine
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(2,6-dimethoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-fluoro-N-[(3-methylphenyl)methyl]-N-(propan-2-yl)-5-sulfamoylbenzamide
N-{5-[(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-1-oxo-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-5-yl]thiophen-2-yl}acetamide
4-[4-(2-propyl-1,3-thiazole-4-carbonyl)piperazine-1-carbonyl]morpholine
8-[4-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinoline
N-[(4-fluorophenyl)methyl]-N-(1-methoxypropan-2-yl)-2,4-dimethyl-1,3-oxazole-5-carboxamide
3-{5-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-(propan-2-yl)propanamide
N-[(1R,3R)-3-aminocyclopentyl]-4-methoxy-3,5-dimethylbenzene-1-sulfonamide
2-(dimethylamino)-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)benzamide
4-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-2-(1-methyl-1H-pyrrol-3-yl)acetamide
2-amino-4-(3-ethyl-1H-pyrazol-5-yl)-6-(3-methyl-1-propyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-(1H-1,3-benzodiazol-2-yl)-N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]acetamide
N-(1-{1-[(4-hydroxy-3,5-dimethylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
4-hydroxy-N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
1-(3,4-dimethoxybenzenesulfonyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-{[4-(difluoromethoxy)phenyl]methyl}-3-(2-methoxybenzoyl)piperidine