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1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]pent-4-en-1-one
1-[4-(naphthalen-2-yl)piperazin-1-yl]-2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethan-1-one
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
N-(2-methylpropyl)-N-[(2E)-3-phenylprop-2-en-1-yl]-2-(pyridin-3-yl)acetamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-[(4-methylphenyl)sulfanyl]propanamide
1-(3-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}(methyl)[1-(pyrimidin-4-yl)ethyl]amine
N-({8-[(2-hydroxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)benzamide
2-[3-(hydroxymethyl)-3-propylpiperidin-1-yl]-N-(2-methylbutan-2-yl)acetamide
1-benzyl-N-(butan-2-yl)-2-methyl-5-(2-methylpropanamido)-1H-1,3-benzodiazole-7-carboxamide
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-N-(1H-indazol-7-yl)-1-methylpyrrolidine-3-carboxamide
3-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[(4-fluorophenyl)methyl]-N-methylbenzamide
4-{[2-(1H-indol-3-yl)ethyl]amino}-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
N-methyl-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-(3-acetamido-4-fluorophenyl)-4-(2-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
1-methyl-4-[4-(thian-4-yl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-(2-methoxyethyl)-9-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{4-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]benzoyl}piperidine
1-[2-(methylsulfanyl)pyrimidin-4-yl]-3-(2-phenylethyl)piperidine-3-carboxylic acid
3-(2-fluoro-4-methoxyphenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-2-(morpholin-3-yl)ethan-1-one
2,6-dimethyl-3-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]-1,4-dihydropyridin-4-one
(1S,3R)-3-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]cyclohexan-1-amine
[(3-{2-[4-(4-fluorobenzoyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
3-(1H-imidazol-2-yl)-1-(5-methyl-4-phenylthiophene-3-carbonyl)piperidine
[(5-ethylpyridin-2-yl)methyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
5-(2H-1,3-benzodioxol-5-yl)-1-methyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-{3-[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]propyl}pyrrolidin-2-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][1-(furan-2-yl)ethyl]methylamine
(1R,2S)-1-{[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}-2,3-dihydro-1H-inden-2-ol
4-{[2-(4-ethoxyphenyl)-1H-imidazol-1-yl]methyl}-1H-indole
1-{2-[4-(2-cyclohexylpyrimidin-5-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
3-(2-amino-1,3-thiazol-4-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
3-(1-methyl-1H-pyrazol-5-yl)-N-[2-(pyridin-3-ylformamido)ethyl]propanamide
methyl 6-[2-(3,4-dichlorophenyl)morpholin-4-yl]pyridine-3-carboxylate
1-(benzyloxy)-8-[3-(3-methoxyphenyl)propanoyl]-1,8-diazaspiro[4.5]decan-2-one
1-{4-[({[4-(hydroxymethyl)oxan-4-yl]methyl}(methyl)amino)methyl]phenyl}imidazolidin-2-one
ethyl 2-{3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-methylpropanamido}acetate
1-(3-methylphenyl)-4-[(trimethylpyrimidin-4-yl)amino]pyrrolidin-2-one
N-(6-hydroxy-6-methylheptan-2-yl)-5-(2-methoxyacetamido)-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
2,4-dimethoxy-N-({2-[3-(2-methoxyacetamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)benzamide
4-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-3-phenyl-1H-pyrazole
1-[(3-methylpyridin-2-yl)methyl]-4-(2,2,6,6-tetramethylpiperidin-4-yl)piperazine
N-[(8-{[4-(propan-2-yl)phenyl]methyl}-1-oxa-8-azaspiro[4.5]decan-2-yl)methyl]oxane-4-carboxamide
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
2,5-dimethyl-N-(2-{5-methyl-4-[(4-phenylbutanamido)methyl]-1,3-oxazol-2-yl}phenyl)furan-3-carboxamide
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl){[4-(pyrimidin-2-yloxy)phenyl]methyl}amine
6-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-(3-methoxyphenyl)-1-(oxane-4-carbonyl)azetidine