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3-(4-methoxy-3,5-dimethylbenzoyl)-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
(3R,4R)-1-(1H-imidazol-2-ylmethyl)-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
2-cyclopropanecarbonyl-8-(3-methyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(7S,9aR)-N-benzyl-8-methyl-7-(2-methylpropyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
N-[(2-chlorophenyl)methyl]-N-(propan-2-yl)-2-(pyridin-3-yl)acetamide
4-[(1-methyl-1H-imidazol-2-yl)methyl]-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
3-(3,4-dimethylphenyl)-1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]propan-1-one
(2S)-N1-(furan-2-ylmethyl)-N2-[3-(1H-pyrazol-1-yl)phenyl]pyrrolidine-1,2-dicarboxamide
1-{[2-(4-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(pyrrolidine-1-carbonyl)piperidine
(2R,6S)-2,6-dimethyl-4-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]morpholine
{1-[(4-ethoxyphenyl)methyl]-3-[(2-fluorophenyl)methyl]piperidin-3-yl}methanol
1-(2-{4-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}ethyl)-1H-pyrazole
(3R)-1-[(8-chloroquinolin-2-yl)methyl]pyrrolidin-3-ol
6-({[3-(2-fluorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}amino)-2-methylheptan-2-ol
9-{[2-(benzyloxy)phenyl]methyl}-1-methyl-1,4,9-triazaspiro[5.5]undecan-5-one
2-(2-chlorophenyl)-N-[(1-hydroxycyclohexyl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
1-[5-({[2-(furan-2-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
ethyl 4-{[4-(2,5-dimethylfuran-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
4-(4-methyl-1H-pyrazol-1-yl)-1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylic acid
1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
(2R,3R,6R)-3-(4-fluorophenyl)-5-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-3-(2-methoxyphenyl)propanamide
2-methyl-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
4-[4-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-methyl-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]-N-(1,2-oxazol-3-ylmethyl)acetamide
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[4-(methylamino)pyrimidin-2-yl]-2,8-diazaspiro[4.5]decan-3-one
1-cyclopropyl-3-{2-[2-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
1-(2-methoxyethyl)-5-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
N-[(1-methylpiperidin-3-yl)methyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)-N-(2-phenylethyl)propanamide
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-[(2,4-dimethylphenyl)methyl]-4-[5-(methanesulfonylmethyl)pyridin-2-yl]piperazine
N-{1-[1-(2-fluorobenzoyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N-methylpyridine-3-carboxamide
3-[(1-cyclopentylpiperidin-4-yl)oxy]-N-[1-(1,3-dimethyl-1H-pyrazol-4-yl)ethyl]benzamide
5-(1-methyl-1H-pyrazol-4-yl)-1,2,3,4-tetrahydroisoquinoline
5-cyclopropyl-N,N-diethyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
1-(2-chloro-3-methoxyphenyl)-3-(2-propoxyethyl)urea
2-chloro-N-ethyl-4-({[2-(2-ethyl-1H-imidazol-1-yl)ethyl]carbamoyl}amino)benzamide
1-ethyl-3-[2-(4-methoxypiperidin-1-yl)-2-oxoethyl]-3-[3-(trifluoromethyl)phenyl]pyrrolidine-2,5-dione
2-[(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxypiperidin-1-yl]-N-(propan-2-yl)pyridine-4-carboxamide
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-(3-fluorophenyl)ethan-1-one
5-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-1-(furan-3-ylmethyl)-4-phenyl-1H-imidazole
4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}phenol
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
N-[2-(2-methyl-1H-indol-1-yl)ethyl]-2-(2-oxopiperidin-1-yl)acetamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N-(3-{[(3-methylphenyl)methyl]sulfanyl}propyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
2-chloro-6-fluoro-N-[1-(pyrimidin-2-yl)piperidin-3-yl]benzamide
4-{[({4-[3-(diethylamino)-2-hydroxypropoxy]-3-methoxyphenyl}methyl)amino]methyl}hepta-1,6-dien-4-ol
N-[(dimethyl-1,3-thiazol-2-yl)methyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide