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2-methyl-9-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecane
1-(azepan-1-yl)-3-(3-{[(3-hydroxypropyl)(methyl)amino]methyl}phenoxy)propan-2-ol
8-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-{1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-4-yl}piperazin-2-one
4-(5,6,7,8-tetrahydroquinoline-3-carbonyl)-1λ6-thiomorpholine-1,1-dione
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
N-[3-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)propyl]pyridin-3-amine
5-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3,3,3-trifluoropropanamide
3-(2-methyl-1H-indol-1-yl)-N-[1-(4-methylpyridin-2-yl)propyl]propanamide
2-(3-methyl-1,2-oxazol-5-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
N-(2,3-dihydroxypropyl)-6-(2,5-dimethylfuran-3-yl)-N,7-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methylazepane
1-({3-[(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]phenyl}methyl)piperidine-3-carboxamide
N-{2-[2-(dimethylamino)-2-(3-methylphenyl)acetamido]ethyl}-2-methylpropanamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}pyridine-3-sulfonamide
8-[1-(1H-imidazol-1-ylmethyl)cyclopropanecarbonyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
7-(cyclohexylmethyl)-2-(furan-3-carbonyl)-2,7-diazaspiro[4.5]decane
3-methoxy-2-(5-methyl-1H-indol-3-yl)pyridin-4-amine
N-({3-methyl-7-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)furan-2-carboxamide
methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl})(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-[(propan-2-yl)amino]pyridine-3-carboxamide
1-(2-methylpropyl)-4-[4-(naphthalen-2-yl)-1H-pyrazol-5-yl]piperidine
N-ethyl-4-fluoro-2-methoxy-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-cyclopentylacetamide
1-methyl-6-(propan-2-yl)-N-{1-[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]ethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-cyclopropyl-4-methoxy-3-{[1-(pyrimidin-2-yl)piperidin-4-yl]oxy}benzamide
N-methyl-N-[2-(2-methylphenyl)-1-[1-(thiophene-2-carbonyl)piperidin-4-yl]ethyl]-2-(1H-pyrazol-1-yl)acetamide
3-[4-(2,5-difluorophenyl)-1H-pyrazol-5-yl]-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
3-methyl-1-propyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-{pyrazolo[1,5-a]pyrimidine-3-carbonyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{4-[4-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)piperidin-1-yl]phenyl}-2H-1,3-benzodioxole-5-carboxamide
5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine
2-(2-methoxyphenyl)-1-[(4-phenyloxan-4-yl)methyl]-1H-imidazole
1-(benzyloxy)-8-cyclopentanecarbonyl-1,8-diazaspiro[4.5]decan-2-one
4-[4-(5,6-dimethylpyrimidin-4-yl)piperazine-1-carbonyl]-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
N-{[2-(3-methylphenyl)-1,3-thiazol-4-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
9-[(2,3-difluoro-6-methoxyphenyl)methyl]-6-oxa-9-azaspiro[4.5]decane
5-[1-(3-fluoro-4-methoxybenzoyl)piperidin-4-yl]-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
N-[(3,4-dimethoxyphenyl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-(pyridin-4-ylmethyl)benzamide
5-ethyl-3-(2-methylprop-2-en-1-yl)-5-{1-[2-(3,4,5-trimethoxyphenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
4-(4-methoxybenzoyl)-2-(2-phenylethyl)morpholine
3-(1H-imidazol-1-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]butan-1-one
1-[1-(2,6-dimethylphenoxy)propan-2-yl]-4-(1,3-thiazol-2-yl)-1H-1,2,3-triazole
N-[1-(4-ethoxy-3-fluorophenyl)ethyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(3S,5R)-1-(4-hydroxy-3-methylbenzoyl)-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-[2-(1,3-thiazol-4-yl)ethyl]pyridin-2-amine
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-4-(azepan-1-yl)-4-oxobutanamide
3-butyl-1-{4-[6-(piperidine-1-carbonyl)pyrazin-2-yl]phenyl}urea
N-{2-[4-(2-fluorophenyl)-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]ethyl}-2-(1H-pyrazol-1-yl)benzamide