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(2R)-3-(benzyloxy)-2-(5-ethyl-4-phenyl-1H-imidazol-1-yl)propan-1-ol
5-({[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}methyl)-2-hydroxybenzoic acid
5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)carbamoyl}amino)-N,N-dimethyl-1-benzothiophene-2-carboxamide
4-(2-hydroxy-3-methylbenzoyl)-1-(4-methylphenyl)piperazin-2-one
[1-(4-ethyl-5-methylpyrimidin-2-yl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
2-(dimethylamino)-2-(3-fluorophenyl)-N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
N-(butan-2-yl)-1-(7-methoxy-4-methylquinazolin-2-yl)piperidine-4-carboxamide
2-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-3,4,7-trimethyl-1H-indole
[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl][1-(1H-imidazol-1-yl)propan-2-yl]amine
3-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
methyl 1-(2-methoxyethyl)-3-(3-methylbutanamido)-5-{[(5-methylfuran-2-yl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-({3-[2-(ethoxymethyl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
2-(dimethylamino)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-(4-fluorophenyl)ethan-1-one
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(4-methoxyphenyl)acetamide
N-cyclobutyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylfuran-2-carboxamide
6-(2,5-dimethylbenzoyl)-1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octane
(2S)-2-acetamido-N-ethyl-4-methyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}pentanamide
2-methyl-3-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,2,3,4-tetrahydroisoquinoline
N-(2-hydroxyethyl)-N-[(5-methylthiophen-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanamide
methyl 3-(naphthalen-2-ylmethyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2,5-dimethyl-3-[4-(oxolan-2-ylmethyl)piperazin-1-yl]pyrazine
[(2S)-1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)pyrrolidin-2-yl]methanol
1-(furan-2-yl)-2-[2-methyl-4-(3-methylphenyl)-5-oxopiperazin-1-yl]ethane-1,2-dione
2-[1-(3-methylbutyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
1-(cyclopropylmethyl)-5-(4-fluorobenzoyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]benzenesulfonamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(4-methoxyphenyl)ethyl]acetamide
4-(4-{[3-(2-hydroxyethyl)-4-[(4-methoxy-3-methylphenyl)methyl]piperazin-1-yl]methyl}phenyl)but-3-yn-1-ol
N-cycloheptyl-3-{methyl[1-(1,2-oxazol-3-yl)ethyl]amino}propanamide
5-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-2-phenyl-1,3-thiazole
1-(3-chlorophenyl)-4-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-2-one
3-(but-3-en-1-yl)-5-[(4-fluorophenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
(3aR,6aR)-2-cyclobutanecarbonyl-5-(3,4-dimethylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[(3-methylpyridin-2-yl)methyl]-4-[(2-phenyl-1H-imidazol-4-yl)methyl]piperazine
methyl 3-[2-(3-fluorophenyl)acetamido]-6-{[(2-methoxyethyl)(propan-2-yl)amino]methyl}thieno[2,3-b]pyridine-2-carboxylate
6-(4-methoxy-3,5-dimethylphenyl)-N,N-dimethylpyridazin-3-amine
4-[3-(phenoxymethyl)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
4-{[4-(5-ethyl-2-methylpyrimidin-4-yl)piperazin-1-yl]methyl}-2,1,3-benzothiadiazole
4-{1-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]piperidin-4-yl}pyridine
benzyl(methyl){[4-(oxolan-2-ylmethyl)-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}amine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[1-(pyrimidin-4-yl)ethyl]piperidine-4-carboxamide
2-{2-[5-(2-methylpropyl)-1,2-oxazole-3-carbonyl]-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-1-yl}pyridine
1-[4-(cyclopentylamino)-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)benzamide
4-(6-methoxypyridin-2-yl)-2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-ylmethyl}phenol
2-methoxy-4-{[5-(morpholin-4-ylmethyl)quinolin-8-yl]oxy}pyridine-3-carbonitrile
ethyl 4-[2-(5-acetylthiophen-3-yl)acetyl]piperazine-1-carboxylate