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1-[1-ethyl-5-(furan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
N-[(2,6-difluorophenyl)methyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
3-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1λ6-thiane-1,1-dione
8-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,3-dioxa-8-azaspiro[4.5]decan-2-one
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
N4-methyl-N4-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrimidine-2,4,6-triamine
N-cyclopropyl-2-(pyridin-4-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-acetyl-8-[2-(4-fluoro-3-methylphenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-(1-benzothiophen-3-yl)-N-[(2,3-dimethoxyphenyl)methyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(2-hydroxyethyl)-N-(1-phenylethyl)-5-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-{5-[1-(2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetyl)piperidin-4-yl]-1H-pyrazol-3-yl}acetic acid
methyl 2-(3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamido)acetate
5-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-5,7-dimethyl-N-[(3S)-2-oxoazepan-3-yl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-methyl-N-[3-(morpholin-4-yl)propyl]acetamide
1-{3-[(3S,4S)-3-hydroxy-4-(piperidin-1-yl)pyrrolidin-1-yl]-3-oxopropyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
ethyl 4-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)butanoate
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
N-cyclopropyl-3-methyl-N-{[5,6,7-trimethoxy-2-(2-methylphenyl)quinolin-3-yl]methyl}thiophene-2-carboxamide
(3S,4R)-3-ethyl-1-[(5-ethylpyridin-2-yl)methyl]-4-methylpiperidin-4-ol
1-[(2,5-difluorophenyl)methyl]-5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)pyrrolidin-2-one
2-(2-methoxyethyl)-4-[4-(4-propylpiperazine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
1-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
(1R,7S)-3-(3-methylbutyl)-6-(3-oxopiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-{[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
N-[4-(2-butoxyacetamido)-2-methoxyphenyl]butanamide
[(4-chloro-3-fluorophenyl)methyl](methyl)(1,2-oxazol-3-ylmethyl)amine
N-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-4-amine
2-[4-hydroxy-2-(pyridin-2-yl)pyrimidine-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]propanamide
2-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}pyridin-3-ol
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-1H-pyrrolo[2,3-b]pyridin-6-amine
2-hydroxy-1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-4-(methylsulfanyl)butan-1-one
methyl 2-(diethylsulfamoyl)-6-[1-(2-methoxyphenyl)propan-2-yl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
ethyl 4-({[(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amino}methyl)-1H-pyrazole-3-carboxylate
[2-(2-ethylphenoxy)ethyl][(2S)-oxolan-2-ylmethyl]amine
1-(azepan-1-yl)-3-(4-methoxyphenyl)-3-phenylpropan-1-one
3-{[7-(1-hydroxy-3-phenylpropyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-6-methyl-4H-chromen-4-one
ethyl 1-{1-[3-(4-fluorobenzenesulfonamido)phenyl]piperidin-4-yl}piperidine-4-carboxylate
(3R,4R)-4-(hydroxymethyl)-1-[2-(2-methylphenyl)benzoyl]piperidin-3-ol
2-(5-{[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]methyl}-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl)acetic acid
3-benzyl-4-(7-chloro-3,5-dimethyl-1-benzofuran-2-carbonyl)piperazin-2-one
N-[2-(3-methoxyphenyl)-1-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-4-yl}ethyl]-N-methyloxane-4-carboxamide
N-[1-(2-chlorophenyl)ethyl]-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanamide
[(3R,4R)-1-[(8-fluoroquinolin-2-yl)methyl]-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
2-(2H-1,2,3-benzotriazol-2-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}acetamide
2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]acetamide
5-[1-({3-methoxy-4-[(3-methylbut-2-en-1-yl)oxy]phenyl}methyl)pyrrolidin-2-yl]-3-methyl-1,2,4-oxadiazole