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N-[(2R,3R)-1'-(3-methoxypropanoyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
2-{[7-(1-benzofuran-5-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
1-methyl-4-{1-[1-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperidin-4-yl]ethyl}piperazine
methyl 2-(azocane-1-sulfonyl)-6-(2-methylpropanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-{[3-(2H-1,3-benzodioxol-5-ylmethoxy)phenyl]methyl}-3-methyl-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
2-methyl-6-{1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}pyrimidin-4-ol
1'-[3-(1H-pyrazol-1-yl)benzoyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
1-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-[3-(5-ethyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
3-{[4-(3-chlorophenyl)-5-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
2-(4-chlorophenyl)-1-[3-(piperidin-1-yl)pyrrolidin-1-yl]ethan-1-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[1-(pyrimidin-4-yl)ethyl]amine
2-(1H-imidazol-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}benzamide
3-(3-benzyl-1H-1,2,4-triazol-5-yl)-1-methyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]urea
(3S,5R)-1-butyl-5-[(pyridin-3-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylacetamide
3-({methyl[(3-methyl-1H-indol-2-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
6-[(2-methylphenyl)methyl]-N-(3-phenylpropyl)-6-azaspiro[2.5]octane-1-carboxamide
5-[1-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-3-yl]-N-[(3,5-dimethoxyphenyl)methyl]-4-methyl-1,3-thiazol-2-amine
3-(2-methoxyethyl)-5-(5-methyl-1-propyl-1H-pyrazol-4-yl)-1,2,4-oxadiazole
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-tert-butylbenzene-1-sulfonamide
3-{2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-oxoethyl}-4-(furan-3-ylmethyl)piperazin-2-one
ethyl 1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-chloro-1-methyl-3-{[(1S,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}-1H-indazole
butyl 2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
2-[8-(1H-indol-3-ylmethyl)-1-(3-methylbutyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetamide
5-{[2-(4-hydroxyphenyl)ethyl]amino}-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
[(3R,4R)-1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
N-(2,1,3-benzoxadiazol-5-ylmethyl)-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-benzyl-3-[5-oxo-2-(thiophen-3-ylmethyl)pyrrolidin-2-yl]propanamide
1-[(2-fluorophenyl)methyl]-N-(oxolan-3-yl)-1H-1,2,3-triazole-4-carboxamide
2-(2-chlorobenzoyl)-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclohexyl-N-methyl-3-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]oxy}benzamide
3-{1-[(3-ethoxy-4-methoxyphenyl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
5-(4-fluorophenyl)-3-[4-(pyrazin-2-yl)piperazin-1-yl]-1,2,4-triazine
3-(2-ethyl-1H-1,3-benzodiazol-6-yl)-1-[1-(pyridin-3-ylmethyl)piperidin-3-yl]urea
2,3-dimethyl-5-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
2-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
6-fluoro-2-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}quinolin-4-ol
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2-(1H-pyrazol-1-yl)acetamide
8-(3-aminopropanoyl)-2-(phenoxymethyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]propanamide
2-(4-{methyl[(3-methylthiophen-2-yl)methyl]amino}pyrimidin-5-yl)acetic acid
1-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)-4-(2-fluorophenyl)piperazine
6-(dimethyl-1,2-oxazole-4-carbonyl)-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide