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2-[(3-methoxyphenyl)methyl]-8-(3,3,3-trifluoropropanoyl)-2,8-diazaspiro[4.5]decan-3-one
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-ethyl-N-methylpyrimidine-5-carboxamide
7-[(6-ethoxyquinolin-2-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
(3S)-N-tert-butyl-2-[3-(1H-pyrazol-4-yl)propanoyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N1-[4-chloro-2-(trifluoromethyl)phenyl]-N3-ethylpyrrolidine-1,3-dicarboxamide
N-[(3R,4R)-3-hydroxy-1-(3-hydroxy-2-methylbenzoyl)piperidin-4-yl]pyridine-2-carboxamide
3-[4-chloro-3-(trifluoromethyl)phenyl]-6-methylpyridazine
2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-1-(morpholin-4-yl)ethan-1-one
(1R,2S,6R,7S)-4-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-azatricyclo[5.2.2.02,6]undecane
2-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-methoxypyridine
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(2-phenylpropyl)piperidin-4-ol
N-cyclobutyl-2-{1-[(3,5-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-imidazole-4-carboxylic acid
4-[2-(1H-indazol-1-yl)acetyl]-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
3-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
N-[(3R,5S)-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
4-[(3-{[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]thiomorpholine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-6-methyl-2-(pyridin-3-yl)pyrimidin-4-amine
1-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
4-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,2-dihydrophthalazin-1-one
1-(4-methanesulfonyl-1,4-diazepan-1-yl)-2-(2-phenyl-1,3-thiazol-4-yl)ethan-1-one
3-chloro-N-[4-(4-{[(3-methyl-1,2-oxazol-5-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)propanamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-1-ethyl-5-(2-methoxyacetamido)-2-(pyridin-3-yl)-1H-1,3-benzodiazole-7-carboxamide
2-{1-[(4-methylphenyl)methyl]-1H-imidazol-2-yl}benzoic acid
N,N-diethyl-1-{5-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
1-(2-{2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-4-methyl-1,2-dihydroquinolin-2-one
2-{1-[(3-chloro-4-methoxyphenyl)methyl]piperidin-2-yl}pyridine
1-[(6-fluoro-1-methyl-1H-indol-3-yl)methyl]-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
9-(7-methyl-1-benzofuran-2-carbonyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[(1R,2S,5R)-6,6-dimethylbicyclo[3.1.1]heptan-2-yl]methyl}-2-(4-methyl-1,4-diazepan-1-yl)acetamide
N-(furan-2-ylmethyl)-4-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carboxamide
4-chloro-N-(2-ethoxypropyl)-N,2-dimethylbenzamide
2-(methylamino)-2-phenyl-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-(2-chlorophenyl)-N-[2-(ethanesulfonyl)ethyl]furan-2-carboxamide
2-(1-benzyl-4-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}piperazin-2-yl)ethan-1-ol
(1R,9S)-5-amino-3-(4-methoxy-3-methylphenyl)-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2-(3-methoxyphenyl)azetidine
5-(2-{2-benzyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxoethyl)imidazolidine-2,4-dione
N-[(2-methylphenyl)methyl]-1-(prop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
9-methoxy-3-[(3-phenoxyphenyl)methyl]-10-(pyrrolidine-1-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepin-7-one
1-cyclohexyl-6-(pyridin-3-ylmethoxy)-4-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1,4-diazepan-2-one
5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]-2-fluorobenzamide
6-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-3-carbonitrile
3-(2-fluorophenyl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-1H-pyrazole-5-carboxamide
N-(1H-imidazol-2-ylmethyl)-1-(4-methoxyphenyl)cyclopentane-1-carboxamide
1-{1-[2-(2-chlorophenoxy)acetyl]piperidin-4-yl}-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
[1-(6-chloro-2-methylquinoline-4-carbonyl)piperidin-2-yl]methanol