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N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)quinoxaline-5-carboxamide
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[(2-methyl-1H-imidazol-4-yl)methyl]-decahydro-1,6-naphthyridin-2-one
5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-(4-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
N-[3-(5-cyclopropyl-1H-pyrazol-1-yl)propyl]-1-(propan-2-yl)piperidine-3-carboxamide
1-[2-hydroxy-3-(4-methoxy-2-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}phenoxy)propyl]piperidin-4-ol
1-{4-[(4-chlorophenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}-2-methylpropan-1-ol
N-{[2-(2-methylphenoxy)pyridin-3-yl]methyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
2-{[(5-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}ethan-1-ol
N-(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
2-(2-aminoacetyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-cyclopentanecarbonyl-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidin-2-amine
2-[(1-{[2-(dimethylamino)ethyl](methyl)amino}hex-5-en-2-yl)oxy]pyridine-4-carbonitrile
N-cyclopropyl-4-methoxy-3-{[1-(3-methylbutyl)piperidin-4-yl]oxy}benzamide
8-methoxy-4-methyl-2-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}quinoline
4-(dimethylamino)-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)benzamide
6-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
N-(2-{7-[(4-fluoro-3-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-[(3-phenylphenyl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
6-(cyclopropylmethoxy)-4-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1-(3-phenylpropyl)-1,4-diazepan-5-one
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-cyclopropyl-2H-1,3-benzodioxole-5-carboxamide
1-(furan-2-carbonyl)-4-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]-1,4-diazepane
N-(cyclopropylmethyl)-2-[1-(4-methoxyphenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetamide
8-[2-(3-fluorophenoxy)acetyl]-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-(1H-pyrazol-1-yl)-1-[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]butan-1-one
2-[5-(3-acetylphenyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]acetic acid
3-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}-2H-chromen-2-one
3-{[1-(1,4-dithiepan-6-yl)piperidin-4-yl]oxy}-N-(2-methoxyethyl)benzamide
1-(4-{[3-(2-hydroxyethyl)-4-(3-phenylpropyl)piperazin-1-yl]methyl}phenyl)imidazolidin-2-one
8-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-benzyl-10-oxo-3,9-diazaspiro[5.6]dodecane-3-sulfonamide
N-(2H-1,3-benzodioxol-5-yl)-6-(3-phenyl-1H-pyrazole-5-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
1-(7-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl)pyrrolidine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-3,5,7-trimethyl-N-(propan-2-yl)-1H-indole-2-carboxamide
3-(2-chlorophenyl)-3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-(2-methoxyethyl)pyrrolidine-2,5-dione
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(4-methylphenyl)propan-1-one
5-(1H-indazole-3-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
methyl 2-(2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-methylacetamido)acetate
3-(azocan-1-ylmethyl)-1-(cyclobutylmethyl)-3-hydroxypiperidin-2-one
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
8-{[4-(azocane-1-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
N-[2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)ethyl]acetamide
4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine
[3-(2-phenoxyethyl)-1-[3-(trifluoromethyl)benzoyl]piperidin-3-yl]methanol
2-{4-[(pyridin-3-ylmethyl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}pyridine-3-carbonitrile
2-(1,2-benzoxazol-3-yl)-N-{2-[1-(propan-2-yl)piperidin-3-yl]ethyl}acetamide
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide