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N-[(3,4-difluorophenyl)methyl]-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]propanamide
ethyl 4-[5-(azepane-1-carbonyl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-amido]piperidine-1-carboxylate
2-{[(4-methylphenyl)methyl]sulfanyl}-N4-(1H-pyrazol-3-ylmethyl)pyrimidine-4,6-diamine
1-(4-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)-1H-1,2,4-triazole
3-{[1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]methyl}benzamide
ethyl 4-{[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}piperidine-1-carboxylate
1-cyclohexyl-3-(cyclopropylmethyl)-N-(oxan-4-yl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-4-methoxypiperidine
2-{2-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
N-[1-(furan-2-ylmethyl)-1H-pyrazol-5-yl]-2-[4-(pyridin-4-yl)-1H-pyrazol-1-yl]acetamide
[(3,5-dichloropyridin-4-yl)methyl](methyl){2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}amine
1-(cyclohexylmethyl)-3-{[(cyclopropylmethyl)amino]methyl}-3-hydroxypiperidin-2-one
2-{4-[4-(piperazin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}quinoxaline
(1R,3S,5S)-3-(4-fluoro-3-methylphenyl)-8-{5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carbonyl}-8-azabicyclo[3.2.1]octane
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
2-[5-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)furan-2-yl]benzonitrile
N-cyclopropyl-N-({4-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-4-methylbenzamide
9-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3,9-diazaspiro[5.6]dodecane
N-{3-[4-(4-methyl-3-phenylpiperazin-1-yl)piperidin-1-yl]phenyl}pyridine-3-carboxamide
3-[2-(2,6-difluorophenyl)ethyl]-1-(1H-imidazol-2-ylmethyl)piperidine
2-{4-[(3,5-difluorophenyl)methyl]-1-[(3,5-dimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
5-acetyl-N-{1-[({2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}carbamoyl)methyl]-1H-pyrazol-4-yl}thiophene-2-carboxamide
1-(dimethylamino)-2-{4-[(2E)-3-[4-(dimethylamino)phenyl]prop-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}propan-2-ol
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
N-(3,4-difluorophenyl)-1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}piperidin-3-amine
dimethyl({4-methyl-5-[1-(quinoxalin-2-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
1-{[5-(1H-imidazol-2-yl)-2,4-dimethylphenyl]methyl}-1H-1,2,4-triazole
(1S,5R)-3-[(2-methyl-1,3-oxazol-4-yl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(1-{[methyl(propan-2-yl)carbamoyl]methyl}piperidin-4-yl)-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
4-{2-[1-(4-chlorophenyl)-5-oxo-3-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl]acetyl}piperazin-2-one
1-({3-[(2-chlorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-4-[1-(pyrrolidin-1-yl)ethyl]piperidine
4-chloro-N-(2-{[(6-hydroxy-1,4-oxazepan-6-yl)methyl]amino}ethyl)benzene-1-sulfonamide
N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidine-6-carboxamide
(1R,2S)-N-tert-butyl-2-(4-acetamidopiperidine-1-carbonyl)cyclohexane-1-carboxamide
(4aR,7aS)-1-(pyrimidin-2-yl)-4-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[1-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
4-[3-(2-benzyl-5-oxopyrrolidin-2-yl)propanoyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
4-hydroxy-3-methyl-N-[1-(3-methylphenyl)-5-oxopyrrolidin-3-yl]benzamide
2-(4-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
3-{[1-(5-propylpyrimidin-4-yl)piperidin-4-yl]amino}azepan-2-one
6-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
N-({8-[(4-ethoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}propan-1-one
1-[(2-methoxyphenyl)methyl]-4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)piperazine
5-acetyl-N-methyl-N-[2-(oxan-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[2-(2-methylphenyl)-2-(4-methylpiperidin-1-yl)ethyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[(1S)-1-{3-[(2-methoxyphenyl)methyl]-1-methyl-1H-1,2,4-triazol-5-yl}-3-(methylsulfanyl)propyl]acetamide
N-{[2-(4-acetylpiperazin-1-yl)-7-methylquinolin-3-yl]methyl}-N-cyclopropyl-3-methylthiophene-2-carboxamide
4-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]benzonitrile
3-methyl-N-[(1S,3S)-3-{[4-(pyridin-2-yl)pyrimidin-2-yl]amino}cyclopentyl]-1H-pyrazole-5-carboxamide