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3-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazole
4-{4-[(2-hydroxy-5-methoxyphenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
10-methoxy-5-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
2-(dimethylamino)-4-methyl-N-[(1-methylpiperidin-4-yl)methyl]-N-(2-phenylethyl)pyrimidine-5-carboxamide
N-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]naphthalene-1-carboxamide
5-(3-fluorophenyl)-3-(3-propoxypiperidin-1-yl)-1,2,4-triazine
N'-(3,5-dimethylphenyl)-N-(1-ethoxy-2-methylpropan-2-yl)propanediamide
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-3-methyl-1H-pyrazole-5-carboxamide
[(1-ethyl-1H-1,3-benzodiazol-2-yl)methyl]({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
N-[(2-methoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-3-(2-methyl-1H-imidazol-1-yl)propanamide
2-{[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
(2S,4S)-N-ethyl-1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-propanamidopyrrolidine-2-carboxamide
N-ethyl-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-4-carboxamide
4-(3-cyclopropyl-5-{7-methylpyrazolo[1,5-a]pyrimidin-6-yl}-1H-1,2,4-triazol-1-yl)-3-methylpyridine
3-[3-(furan-2-yl)-5-[2-(2-oxopiperidin-1-yl)ethyl]-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-[2-methyl-1-(5-methyl-1H-1,3-benzodiazol-2-yl)propyl]pyridine-4-carboxamide
N-[2-(pyridin-4-yl)ethyl]-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-(2-{[1-(9H-purin-6-yl)piperidin-4-yl]amino}ethyl)-1,3-oxazinan-2-one
2-methyl-N-[(5-methylpyrazin-2-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
4-(2-methoxyphenoxy)-1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)piperidine-4-carboxylic acid
3,3-dimethyl-1-[(3S,4R)-4-(propan-2-yl)-1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-3-yl]urea
3-fluoro-N-[(2R,3R)-1'-(1H-imidazol-4-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
1-(1-ethyl-5-methyl-1H-pyrazole-3-carbonyl)-4-(2-methylphenyl)-1,4-diazepane
3-[methyl({2-[4-(3-methylphenoxy)piperidin-1-yl]-2-oxoethyl})amino]-1λ6-thiolane-1,1-dione
6-[(4-chlorophenyl)methyl]-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
6-{3-oxo-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-9-yl}pyridine-3-carboxylic acid
(2R,3R,6R)-3-(4-methoxyphenyl)-5-(1,3-thiazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-{2-[methyl(2-methylpropyl)amino]ethyl}-8-[(2R)-oxolane-2-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3S,4S)-4-(pyrrolidin-1-yl)-1-(quinolin-2-ylmethyl)pyrrolidin-3-ol
N-[(5-methylpyrazin-2-yl)methyl]-1-benzothiophene-5-carboxamide
1-[4-(4-methoxybenzoyl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[1-(1H-1,3-benzodiazol-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-{[4-(3-chlorophenyl)-5-(1-methoxypropyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(3S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
methyl 5-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}-3-cyclobutaneamido-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-cyclohexyl-3-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidine-1-carboxamide
4-[2-(morpholin-4-ylmethyl)phenyl]pyridin-2-amine
(3S,4S)-4-cyclopropyl-1-{[2-(2-fluorophenyl)ethyl]carbamoyl}pyrrolidine-3-carboxylic acid
(2S,4R)-N-(diphenylmethyl)-1-(3-phenylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
1-[(4-fluorophenyl)methyl]-5-(2-methoxyacetamido)-N-[(4-methylphenyl)methyl]-1H-1,3-benzodiazole-7-carboxamide
N-[2-(4-{[3-(1H-indol-3-yl)propanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-[4-(4-fluorophenyl)piperazin-1-yl]ethan-1-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
[(2R)-1-({1-[1-(thiophene-2-carbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)pyrrolidin-2-yl]methanol
ethyl 4-({[5-(2-chloroprop-2-en-1-yl)-6-oxo-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}amino)piperidine-1-carboxylate
N-[(1-methylpiperidin-4-yl)methyl]-4-oxo-N-(2-phenylethyl)-4H-chromene-2-carboxamide
N-[3-(1H-indol-2-yl)phenyl]-1-(2-methylpropanoyl)piperidine-3-carboxamide
1-(5-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-1-methyl-1H-pyrrol-3-yl)ethan-1-one
2-[1-(cyclohexylmethyl)piperazin-2-yl]ethan-1-ol