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N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[3-(naphthalene-1-carbonyl)piperidin-1-yl]-3-(pyridin-2-yl)propan-1-one
5-(5-ethyl-1,3-oxazol-4-yl)-3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazole
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
5-{[2-(methoxymethyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
3-(oxolan-2-ylmethyl)-5-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
3-[4-(ethanesulfonyl)piperazine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole
N-(1-{7-[(3,4-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
2-(4-methoxyphenoxy)-N-{[5-(5-methylpyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
3-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
N-{[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,1-benzoxazole-3-carboxamide
1-(2-methoxyphenyl)-4-[1-oxo-1-(piperidin-1-yl)propan-2-yl]piperazin-2-one
1-{1-[5-(1-ethyl-3-methyl-1H-1,2,4-triazol-5-yl)furan-2-yl]ethyl}piperidine
ethyl 1-(2-chlorophenyl)-5-({[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
N-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-methylacetamide
2-(2,3-dihydro-1H-indol-1-yl)-2-oxo-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
4-ethyl-N-(2-hydroxy-3-methoxypropyl)-N,5-dimethylpyrimidin-2-amine
6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
1-{[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}azepan-2-one
(1S,5R)-6-benzyl-3-(6-methoxypyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 6-(3-cyclohexylpropanoyl)-2-(phenylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-methyl-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-5-(propan-2-yl)-1H-pyrazole-4-carboxamide
4-[1-(2-phenylethyl)pyrrolidin-3-yl]-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidine
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
3-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydroquinolin-2-one
3-[3-(3,4-dimethoxybenzoyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-[(3,5-dimethoxyphenyl)methyl]-3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[(2,3-dimethyl-1H-indol-7-yl)methyl]-N,N-dimethylpiperazine-1-sulfonamide
2-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-phenylpropanamide
3-benzyl-4-[3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanoyl]piperazin-2-one
2-(4-methoxy-2,5-dimethylphenyl)-1-(2,2,2-trifluoroethyl)-1H-imidazole
2-amino-4-methyl-N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]pyrimidine-5-carboxamide
methyl 3-[({7-chloro-5-[2-(methylsulfanyl)pyrimidin-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methyl)carbamoyl]benzoate
methyl 2-{3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}butanoate
2-[1-(cyclohexylmethyl)-3-oxopiperazin-2-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
4-(4-chlorophenoxy)-1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-ethyl-4-(hydroxymethyl)-N-[(2E)-3-phenylprop-2-en-1-yl]benzamide
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
7-fluoro-3-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1-benzofuran-2-carboxamide
1-methyl-6-(2-phenylethyl)-N-[1-(pyrimidin-4-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(1S,4S)-2-(3-chlorophenyl)-5-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-5-propyl-1,3,4-oxadiazol-2-amine
3-[1-(4-methanesulfonylphenyl)-3,5-dimethyl-1H-pyrazol-4-yl]propanoic acid
1-(2-{4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-4-yl)piperidin-4-ol
ethyl 4-[(4-methoxyphenyl)methyl]-1-(pyridine-3-sulfonyl)piperidine-4-carboxylate
3-[3-(2-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-1H-imidazol-1-yl)phenyl]-1,3-oxazolidin-2-one
5-(2-{[(2-fluorophenyl)methyl]amino}ethyl)-1-[3-(methylsulfanyl)propyl]pyrrolidin-2-one
3-(2-oxo-2-{3-propyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethyl)-2,3-dihydro-1λ6-thiophene-1,1-dione
N-(1-{1-[3-(5-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide