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(1R,3S)-3-(2-aminoethoxy)-7-(4-ethyl-1,2,3-thiadiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
[4-(2-phenylethyl)-1-[(2,3,6-trifluorophenyl)methyl]piperidin-4-yl]methanol
methyl[(3-{[1-(4-methylbenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](thiophen-3-ylmethyl)amine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(6-methylpyridazin-3-yl)-6-(morpholin-4-yl)-decahydroisoquinoline
3-(1H-indol-3-yl)-1-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}propan-1-one
1-(4-phenylbutanoyl)-4-propyl-1,4-diazepan-5-one
4-methoxy-3-{1-[2-(propan-2-ylsulfanyl)ethyl]-1H-1,2,3-triazol-4-yl}phenol
N-[(3R,4S)-1-methanesulfonyl-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]cyclopentanecarboxamide
N-{2-[(4-methylpyridin-2-yl)amino]ethyl}-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-ethyl-5-hydroxy-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)adamantane-1-carboxamide
6-hydroxy-1-(pyridin-3-ylmethyl)-4-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-diazepan-2-one
6,7-dimethoxy-2-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-3-yl}-1,2,3,4-tetrahydroisoquinoline
N-[4-(3-fluorophenyl)phenyl]-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carboxamide
2-acetyl-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}quinolin-8-ol
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(propan-2-yl)-N-(pyridin-3-ylmethyl)quinoline-4-carboxamide
N-[4-(3-methanesulfonamidopropanamido)phenyl]-5-methylfuran-2-carboxamide
[(1-benzyl-1H-imidazol-2-yl)methyl](methyl){[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
1-[(3,5-dimethylphenyl)methyl]-4-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperazin-2-one
[2-(3-methoxyphenyl)ethyl]({[7-(methylsulfanyl)-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
1-[5-(methanesulfonylmethyl)pyridin-2-yl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
3-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-4H-chromen-4-one
(2R,4R)-N-[2-(2,4-dichlorophenyl)ethyl]-4-hydroxypyrrolidine-2-carboxamide
1-{1'-[2-(4,5-dimethyl-1H-imidazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-methylfuran-2-carboxamide
2-{6-hydroxy-4-[4-methyl-6-(methylamino)pyrimidin-2-yl]-1,4-diazepan-1-yl}-N-methylacetamide
8-(5-hydroxypyrazine-2-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
N-[(4-chlorophenyl)methyl]-1-(4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-1-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]propan-1-one
N-(2,3-dihydro-1H-inden-2-yl)-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(benzylsulfamoyl)({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl})amine
(3S,4S)-3-hydroxy-4-[methyl({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amino]-1λ6-thiolane-1,1-dione
1'-[(2-ethylpyrimidin-5-yl)methyl]spiro[indene-1,4'-piperidine]
4-(1H-pyrazol-1-yl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidine-4-carboxylic acid
(2R,3R,6R)-5-(dimethyl-1,2-oxazole-4-carbonyl)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(oxolan-2-ylmethyl)-5-{1-[3-(prop-2-en-1-yloxy)benzoyl]piperidin-4-yl}-5-propylimidazolidine-2,4-dione
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,5-diazatricyclo[5.2.2.02,6]undecane
methyl (2S,4R)-1-methyl-4-(1,8-naphthyridine-2-amido)pyrrolidine-2-carboxylate
2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
2-methyl-5-(propan-2-yl)-N-{[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]methyl}furan-3-carboxamide
1-(5-chloro-2-methoxybenzoyl)-3-(2-methoxyphenoxy)azetidine
{[2-methanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)(quinolin-4-ylmethyl)amine
1-(5-methanesulfonyl-2-methylphenyl)-3-[(1-propyl-1H-pyrazol-4-yl)methyl]urea
N-{2-[(E)-2-(8-hydroxyquinolin-2-yl)ethenyl]phenyl}-2,4-dimethyl-1,3-oxazole-5-carboxamide
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(4-fluorophenyl)methyl]piperazin-2-one
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(5-methylhexan-2-yl)piperidine
8-(pyrrolidine-1-sulfonyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid