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3-butanamido-N-(2-hydroxy-3-phenylpropyl)-4-methylbenzamide
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-3-(3-methyl-1H-pyrazol-1-yl)propanamide
N-[3-(furan-2-yl)propyl]-2-(5-oxo-1-phenyl-3-propyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
(2S,4R)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-1-[(3-methoxyphenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
3-{1-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-3-yl}-N,N-dimethylpropanamide
2-(1-methyl-4-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}piperazin-2-yl)ethan-1-ol
4-[5-(1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}pyrrolidin-2-yl)-1,2,4-oxadiazol-3-yl]pyridine
4-{[1-(2-fluorophenyl)-5-(1H-1,2,3,4-tetrazol-1-ylmethyl)-1H-1,2,4-triazol-3-yl]methyl}-1-methylpiperidine
6-[8-(3-methylbutyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
1-(2-methoxyethyl)-5-(2-methylpiperidine-1-carbonyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
N-[4-(1H-indol-2-yl)phenyl]-1-(3-methoxypropanoyl)piperidine-4-carboxamide
1-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(pyridin-3-ylmethyl)spiro[2.4]heptane-1-carboxamide
[(3R,4R)-1-(3-chloropyridin-2-yl)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
7-methyl-2-(1-methyl-1H-pyrazol-4-yl)-N-(1,1,1-trifluoropropan-2-yl)quinoline-4-carboxamide
1-(2-chlorophenyl)-4-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-5-methylpiperazin-2-one
N-{[2-(morpholin-4-yl)-1,3-thiazol-5-yl]methyl}-1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
5-benzoyl-1-(2-methylpropyl)-N-(pyridin-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1-benzothiophen-2-ylmethyl)({4-[(1-cyclohexanecarbonylpiperidin-4-yl)oxy]phenyl}methyl)methylamine
7-(cyclopropylmethyl)-6-(2-fluoro-4-methoxyphenyl)-N,N-dimethyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-(1H-imidazol-1-yl)-1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]propan-1-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}quinoxaline-5-carboxamide
ethyl 1-(4-ethenylbenzoyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[2-(3-chlorophenyl)ethyl]-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-oxo-1H,2H,5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
5-{1-[2-(3,5-difluorophenyl)acetyl]piperidin-4-yl}-5-ethyl-3-(2-methylprop-2-en-1-yl)imidazolidine-2,4-dione
N-[2-chloro-5-(diethylcarbamoyl)phenyl]-2-methyloxolane-2-carboxamide
2-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridin-6-yl]-N-[2-(4-methoxyphenyl)ethyl]acetamide
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
(1S,4S)-2-(2H-1,3-benzodioxol-5-yl)-5-[(2,4-dimethoxy-3-methylphenyl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-[4-(aminomethyl)piperidin-1-yl]-2-(oxan-2-ylmethyl)-2,3-dihydropyridazin-3-one
3-[4-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
2-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}acetamide
1-[3-(1H-imidazol-1-yl)propyl]-4-(2-phenylpropyl)-1H-1,2,3-triazole
4-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
4-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(4-fluorophenyl)methyl]piperazin-2-one
N-methyl-2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethane-1-sulfonamide
methyl 4-(4-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}piperazin-1-yl)benzoate
1-(benzenesulfonyl)-4-(4-propyl-1H-1,2,3-triazol-1-yl)piperidine
2-butyl-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-1,3-benzoxazole-5-carboxamide
4-{[1-(2-phenylbenzoyl)piperidin-2-yl]methyl}morpholine
3-[4-(aminomethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
4-(4-amino-5-methylpyrimidin-2-yl)-1-[(4-fluorophenyl)methyl]piperazin-2-one
4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]-1-[(2R)-oxolane-2-carbonyl]piperidine
1-[3-(3-methylbenzamido)phenyl]-5-oxopyrrolidine-3-carboxylic acid
N-[(2,3-dimethylphenyl)methyl]-5-(3-fluorophenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide