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5-[4-(4-methoxyphenyl)-3,3-dimethylpiperazine-1-carbonyl]pyridine-2,4-diol
2-{3-[1-(cyclopropylmethyl)-1H-pyrazol-3-yl]phenyl}pyridine-4-carbonitrile
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-(oxolan-2-ylmethyl)piperidine-4-carboxamide
2-methoxy-N-[(2R,3R)-2-methoxy-1'-(1,3-thiazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
3-(4-methyl-1,3-thiazol-5-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]propan-1-one
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
3-(3-hydroxy-1,2-oxazol-5-yl)-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}propan-1-one
N-(adamantan-1-yl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-[(6-cyclopropylpyrimidin-4-yl)amino]-1-(4-fluorophenyl)pyrrolidin-2-one
2,4-dichloro-3-{[3-(morpholin-4-yl)azetidin-1-yl]methyl}phenol
methyl 1-({4-[3-(thiophen-3-yl)-1H-pyrazole-5-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-4-(4-methoxyphenoxy)piperidine
1-[(3-fluorophenyl)methyl]-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]-6-oxopiperidine-3-carboxamide
3-(1-methyl-1H-pyrazol-4-yl)-1-(1,2,3,4-tetrahydronaphthalen-2-yl)urea
1-[4-(ethylsulfanyl)phenyl]-3-(1-hydroxybutan-2-yl)-3-(pyridin-4-ylmethyl)urea
(3S,4S)-1-[3-(dimethylsulfamoyl)propyl]-4-propylpyrrolidine-3-carboxylic acid
4-fluoro-N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]benzamide
2-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-(2-chloro-5-sulfamoylphenyl)-3-[3-(2-oxopyrrolidin-1-yl)propyl]urea
1-(4-benzylpiperazin-1-yl)-3-{1-[(2-methylphenyl)methyl]piperidin-3-yl}propan-1-one
1-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazole
1-(2-ethoxyphenyl)-4-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperazine
(3R,5S)-5-{3-[(4-methoxyphenyl)methyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl}pyrrolidin-3-ol
(2S)-4-methyl-2-phenyl-1-[(2,3,4-trimethoxyphenyl)methyl]piperazine
2-{[3-(pyridine-3-carbonyl)piperidin-1-yl]methyl}quinolin-4-ol
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,6-dichlorophenyl)urea
(2S,4R)-N-(1-benzothiophen-2-ylmethyl)-1-[(2-chloro-6-fluorophenyl)methyl]-N-methyl-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
4-(4-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-1-yl)-2-(pyridin-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(1-{7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclopropanecarboxamide
N-[(6-methylpyridin-2-yl)methyl]-6-[4-(1H-pyrazol-1-yl)benzoyl]-6-azaspiro[2.5]octane-1-carboxamide
1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(thiophen-3-yl)propan-1-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
{4-[(3-fluorophenyl)methyl]-1-[(3-methylquinoxalin-2-yl)methyl]piperidin-4-yl}methanol
4-(furan-3-carbonyl)-9-methoxy-7-(4-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclopentyl-4-oxo-4-(4-phenylazepan-1-yl)butanamide
(3aR,6aR)-2-[(2-chlorophenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(4-{3-[2-methyl-5-(3-methylphenyl)pyrimidin-4-yl]piperidine-1-carbonyl}phenyl)morpholine
5-{2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
N-(2-hydroxyethyl)-3-{5-[1-(propan-2-yl)piperidin-4-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
4-[(2,3-difluoro-6-methoxyphenyl)methyl]-2-ethyl-1-(propan-2-yl)piperazine
1-cyclohexyl-4-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1,4-diazepane
N,N,4-trimethyl-3-({[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
5-oxo-1-(pyridin-4-ylmethyl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-3-carboxamide
2-(1-{[1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
N-[1-(7-{[5-(2-chlorophenyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]-2-methylbenzamide
methyl 1-[(3R,5S)-1-[(3-chlorophenyl)methyl]-5-(4-phenylpiperazine-1-carbonyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-2-hydroxy-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(4-ethoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(1-{1-[4-(2-methylpropyl)benzoyl]piperidin-3-yl}piperidin-4-yl)methanol