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6-[2-(4-chloro-2-methylphenoxy)propanoyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
7-[ethoxy(phenyl)methyl]-4-(1H-indole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-cyclobutyl-2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}acetamide
5-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-N-phenylpyrimidin-2-amine
1-[2-hydroxy-3-(3-{[3-(pyridin-2-yl)azetidin-1-yl]methyl}phenoxy)propyl]piperidin-4-ol
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N2,N4-dimethyl-N2-[3-(oxolan-2-yl)propyl]pyrimidine-2,4-diamine
2-(1H-imidazol-2-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylbenzamide
{1-[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-3-yl}methanol
1-[(3-cyclopropyl-1-propyl-1H-1,2,4-triazol-5-yl)methyl]-1H-indole
4-cyclobutyl-N,6-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyrimidin-2-amine
(3S)-1-[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-ol
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(1-methyl-1H-1,3-benzodiazol-5-yl)urea
2-ethyl-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-5-carboxamide
2-(1-{[4-(piperidine-1-carbonyl)phenyl]methyl}-1H-imidazol-2-yl)benzoic acid
N-methyl-2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[(2E)-3-phenylprop-2-en-1-yl]acetamide
5-(2-methoxyacetamido)-1-methyl-N-(1-phenylcyclopropyl)-2-(pyridin-4-yl)-1H-1,3-benzodiazole-7-carboxamide
3-[(2,3-difluorophenyl)methyl]-1-(2-methoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-(benzenesulfonyl)-3-(3-methylthiophene-2-carbonyl)piperidine
(3S,4R)-1-[3-(dimethylamino)benzoyl]-4-(4-methoxyphenyl)-N,N-dimethylpyrrolidin-3-amine
N,N-dimethyl-5-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1,3-thiazol-2-amine
(5-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}furan-2-yl)methanol
N-benzyl-6-[2-(2-methoxyphenyl)acetyl]-6-azaspiro[2.5]octane-1-carboxamide
3-(1H-pyrazol-5-yl)-1-(1H-pyrrole-2-carbonyl)piperidine
[3-(methylsulfanyl)propyl](3-phenylprop-2-yn-1-yl)(prop-2-en-1-yl)amine
2-(dimethyl-1,2-oxazol-4-yl)-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)acetamide
9-[2-(benzyloxy)acetyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-N-ethyl-4-[2-(3-hydroxyphenyl)acetamido]-1-[(3E)-pent-3-enoyl]pyrrolidine-2-carboxamide
N-[3-(furan-2-yl)propyl]-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
N-[2-(1-benzylpiperidin-4-yl)ethyl]oxane-2-carboxamide
N-[(2R,3R)-2-methoxy-1'-propyl-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
2-(azepan-1-yl)-1-[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-[(3,4-dimethoxyphenyl)methyl]-3-(3-fluorophenyl)-N-(pyridin-2-ylmethyl)benzamide
2-(dimethylamino)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
1-[(4aS,8aR)-decahydroisoquinolin-2-yl]-3-[5-(3-phenylpropyl)-1,3,4-oxadiazol-2-yl]propan-1-one
(3R,5S)-N-[2-(1H-imidazol-4-yl)ethyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-[3-(trifluoromethyl)phenoxymethyl]piperidine-3-carboxamide
3-[(3R,4S)-1-(4-ethylbenzoyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
3-(1H-imidazol-2-yl)-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
1,4-dimethyl-9-[(2,4,5-trimethylphenyl)methyl]-1,4,9-triazaspiro[5.5]undecane
1-benzyl-3-methyl-8-{[4-(2-methylphenyl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1H-pyrazole-3-carboxamide
4-[(1-acetylpiperidin-4-yl)oxy]-N-(3-ethoxypropyl)-3-methoxybenzamide
4-[3-(2-chlorophenyl)propanoyl]-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(2-phenoxyethyl)piperazine
({1-[2-(4-fluorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
1-[4-({[3-(dimethylamino)-2,2-dimethylpropyl]amino}methyl)-2-methoxyphenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
2-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]morpholine
4-methyl-N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,3-oxazole-5-carboxamide
methyl (2S,4S,5R)-2-ethyl-5-(4-methoxyphenyl)-1-methyl-4-(pyrrolidine-1-carbonyl)pyrrolidine-2-carboxylate