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1-methyl-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[3-(4-fluorophenyl)phenyl]-1-(1-methylcyclopropanecarbonyl)piperidine-3-carboxamide
4-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-1-(thian-4-yl)piperidine
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methylpyridin-4-yl)methyl]acetamide
8-{[2-(benzylamino)pyrimidin-5-yl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
5-(1H-imidazol-1-ylmethyl)-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]furan-2-carboxamide
7-(3,5-difluoropyridine-2-carbonyl)-N-(propan-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(5-ethylfuran-2-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-amine
2-cyclopentanecarbonyl-7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane
1-{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}-4-fluoropiperidine
N-cyclopentyl-2-{4-[3-(furan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}propanamide
N-methyl-5-(morpholin-4-ylmethyl)-N-[2-(phenylsulfanyl)ethyl]furan-3-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-(hydroxymethyl)-5-methyl-1,2-oxazole-3-carboxamide
3-[(cyclooctylamino)methyl]-5,6,7-trimethoxy-N,N-dimethylquinolin-2-amine
N-cyclopentyl-5-(2-methoxyacetyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-(oxolane-3-carbonyl)-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-amine
2-amino-1-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
4-[5-(propan-2-yl)-1H-1,2,4-triazol-3-yl]-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(methylsulfanyl)-N-[5-oxo-1-(2-phenylethyl)pyrrolidin-3-yl]acetamide
3-({1-[2-methyl-2-(morpholin-4-yl)propyl]pyrrolidin-3-yl}methyl)benzoic acid
N-(5-acetyl-2-methoxyphenyl)-4-(morpholin-4-yl)piperidine-1-carboxamide
[(2,5-difluorophenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
methyl 3-(4-methylbenzoyl)-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl({[1-(2-methylpropyl)-2-(oxolan-2-ylmethanesulfonyl)-1H-imidazol-5-yl]methyl})[2-(piperidin-1-yl)ethyl]amine
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
methyl 3-[(2-fluoro-5-methoxyphenyl)methyl]-7-oxo-9-(pyridin-4-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-methyl-3-{1-[1-(propan-2-yl)-1H-pyrazol-4-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazole
4-methoxy-1-[(2S)-2-phenylbutyl]piperidine
6-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]pyrazine-2-carboxylic acid
1-{[3-cyclopentyl-1-(4-methoxyphenyl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-3-ol
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-5-(2-methylpropyl)-1,2-oxazole-3-carboxamide
1-propyl-5-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-benzyl-3-(2-{methyl[2-(pyridin-2-yl)ethyl]carbamoyl}ethyl)piperidine-1-carboxamide
(2S)-N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-hydroxy-3-phenylpropanamide
(2R,3R)-3-{[(2-methoxyphenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
5,6-dimethyl-2-oxo-N-[1-phenyl-2-(1H-pyrazol-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N-[(3-methylthiophen-2-yl)methyl]-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
2-{4-methyl-6-[3-(5-methyl-1,2,4-oxadiazol-3-yl)piperidin-1-yl]pyrimidin-2-yl}phenol
4-{2-[2-(3-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-(1-methylpiperidine-2-carbonyl)piperidine
N-[(3-methoxyphenyl)methyl]-3-methyl-N-(prop-2-en-1-yl)furan-2-carboxamide
N-[1-(1-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
N-[(3S,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(3aR,6aR)-2-(2-hydroxyethyl)-5-(morpholine-4-sulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2,2-dimethyloxane-4-carboxamide
3-(benzyloxy)-1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
3-(but-2-yn-1-yl)-5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-(3-phenylpropyl)imidazolidine-2,4-dione
[(3R,4R)-1-(2,6-difluorobenzoyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
[(3R,4R)-4-[(dimethylamino)methyl]-1-[(2-ethylphenyl)methyl]pyrrolidin-3-yl]methanol
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1-methylpiperidin-4-amine
1-(4-methyl-1,2,5-oxadiazol-3-yl)-4-{[5-methyl-2-(4-phenylphenyl)-1,3-oxazol-4-yl]methyl}piperazine