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5-ethyl-5-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
4-[3-(5-methylthiophen-2-yl)-5-(morpholine-4-sulfonyl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-[2-(5-methyl-1,2,4-oxadiazol-3-yl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-(cyclopropylmethyl)-2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-(1,2-oxazol-3-ylmethyl)-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-3-[4-(trifluoromethoxy)phenyl]benzamide
3-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-1H-pyrazole
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-ol
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
1-[2-(3-chlorophenyl)ethyl]-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}pyrrolidin-2-one
2-[5-(5-ethyl-1,2-oxazol-3-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]-6-methylpyridine
dimethyl(3-{2-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
(2,3-dihydro-1-benzofuran-5-ylmethyl)[2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(pyridin-2-ylmethyl)-decahydroisoquinoline
2-{[(5-ethyl-2-methylpyrimidin-4-yl)(methyl)amino]methyl}-3H,4H-thieno[3,2-d]pyrimidin-4-one
3-[3-(4-fluorophenyl)phenyl]-1-methyl-1-(piperidin-4-yl)urea
1-[4-(propan-2-yl)-1,3-thiazole-2-carbonyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-cyclopropyl-2-(dimethylamino)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-methylphenyl)acetamide
3-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1,6-dimethyl-1,4-dihydroquinolin-4-one
3-({3-[3-(pyrimidin-5-yl)phenyl]-1H-pyrazol-1-yl}methyl)benzonitrile
(3R,4R)-1-[(2-hydroxy-5-methoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbenzamide
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[(1-cyclopentylpiperidin-4-yl)methyl]-N-(oxolan-2-ylmethyl)acetamide
4-[(2-methoxyphenyl)methyl]-11-{[(5-phenyl-1,2-oxazol-3-yl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
3-{2-[8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-ethyl-4-[5-(3-phenoxypropanamido)-1H-pyrazol-1-yl]piperidine-1-carboxamide
methyl 3-(furan-2-amido)-1-(2-methoxyethyl)-5-[(2-phenylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-(2-{[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]amino}ethyl)methanesulfonamide
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-fluorophenoxy)piperidine
N-(2,3-dihydro-1H-inden-2-yl)-3-(3-hydroxy-3-methylbutyl)benzamide
2-butyl-4-{[3-(2-chlorophenoxy)azetidin-1-yl]methyl}-1H-imidazole
1-(adamantan-1-yl)-3-[2-(4-ethylmorpholin-2-yl)ethyl]urea
2-methyl-6-({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}amino)heptan-2-ol
2-(3-{[(1R,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}phenoxy)acetamide
2-amino-4-(5-cyano-1-methyl-1H-pyrrol-3-yl)-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
(4aS,8aR)-1-(2-phenylethyl)-6-(pyridin-3-ylmethyl)-decahydro-1,6-naphthyridin-2-one
2-(2,3-dihydro-1H-isoindole-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]quinoline-2-carboxamide
N,N-dimethyl-6-[2-(pyridin-2-yl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
1-[(2,5-dimethoxyphenyl)methyl]-3-(3-methyl-1,2,4-thiadiazol-5-yl)urea
2-methyl-N-({1-[(4-methylpiperazin-1-yl)methyl]cyclopropyl}methyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]ethan-1-one
1-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-4-[(4-fluorophenyl)methyl]piperidine
4-{[4-(2-methoxyacetyl)-1,4-diazepan-1-yl]methyl}-N-(1-methyl-1H-pyrazol-4-yl)benzamide
(2S,4S)-4-{[(3,4-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(propan-2-yl)pyrrolidine-2-carboxamide
1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)piperidine-3-carboxamide
2-(oxolan-2-ylmethyl)-9-{[4-(propan-2-yl)phenyl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
2-{4-[(4-fluorophenyl)methyl]-3-oxopiperazin-1-yl}-2-(3-hydroxyphenyl)acetic acid
1-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(pyridin-3-yl)ethan-1-one