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N-(2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-oxoethyl)acetamide
1-(cyclohexylmethyl)-4-(quinolin-6-yloxy)piperidine-4-carboxylic acid
4-(4-{4-[(3-methylpiperidin-1-yl)methyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)pyrimidin-2-amine
6-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pyridine-3-carbonitrile
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1H-pyrazol-4-yl)ethyl]amine
methyl 1-[(3R,5S)-5-[(diphenylmethyl)carbamoyl]-1-[(2-ethoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(phenylformamido)acetamide
4-hydroxy-2-(4-methylphenyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)pyrimidine-5-carboxamide
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(5-methyl-1,3-oxazole-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-{1-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-2-phenylethyl}-N-methylthiophene-2-carboxamide
1-[(3R,4R)-3-(hydroxymethyl)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}pyrrolidin-1-yl]-3-phenylpropan-1-one
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-(propan-2-yl)pyridine-4-carboxamide
N-{[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-phenylacetamide
N,N-dimethyl-7-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-(4-chlorophenyl)-5-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}pyrimidine
6-{[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]amino}-N,N-dimethylpyridine-3-carboxamide
9-(3-hydroxypropanoyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2-chloro-4-fluorophenyl)-N-{[8-methyl-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}acetamide
N-(cyclopropylmethyl)-2-methyl-N-(oxolan-2-ylmethyl)-3-[(pyridin-3-ylmethyl)amino]benzamide
N-ethyl-3-methyl-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
3-ethyl-6-[3-(morpholin-4-yl)azetidine-1-carbonyl]-3H-imidazo[4,5-b]pyridin-2-amine
1-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-4-(piperidin-1-yl)piperidine-4-carboxamide
N-cyclopropyl-3-{[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]sulfamoyl}benzamide
N-(1-{1-[(3-ethoxy-2-hydroxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N-methylthiophene-2-carboxamide
1-(3-{5-methoxy-1-oxa-9-azaspiro[5.5]undecane-9-carbonyl}phenyl)imidazolidin-2-one
2-{2-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]-4-(pyrazin-2-yl)phenoxy}acetic acid
(4aS,8aR)-6-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-decahydro-1,6-naphthyridine-4a-carboxylic acid
3,3-dimethyl-1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-4-(morpholin-4-ylmethyl)piperidin-4-ol
[(2,5-dimethylphenyl)methyl](methyl){[5-(methylsulfanyl)-4-(oxolan-2-ylmethyl)-4H-1,2,4-triazol-3-yl]methyl}amine
3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1H-1,2,4-triazole
2-[(3R,4S)-3-(2-cyclopentylacetamido)-4-cyclopropylpyrrolidin-1-yl]pyridine-3-carboxamide
1-benzyl-8-[(2-chloro-6-fluorophenyl)methyl]-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-{3-[ethyl(methyl)amino]-2-methylpropanoyl}-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(propan-2-yloxy)ethan-1-one
1-(4-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
2-{1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl}benzoic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-3-(3-methoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
4-[6-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridazin-3-yl]thiomorpholine
N-[(1-cyclopentylpiperidin-4-yl)methyl]-4-methyl-N-(pyridin-3-ylmethyl)pyrimidine-5-carboxamide
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-1,2,4-triazol-1-yl)butan-1-one
(4aS,8aS)-2-(1H-pyrazole-4-carbonyl)-decahydroisoquinolin-4a-ol
2-(2-phenylethyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1,3-benzoxazole-5-carboxamide
(4aR,8aR)-4-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydro-2H-1,4-benzoxazine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(2-methoxyphenyl)ethan-1-one
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
2-(2-aminoethyl)-N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}quinazolin-4-amine
4-[3-(ethoxycarbonyl)-3-[(3-methoxyphenyl)methyl]piperidine-1-carbonyl]pyridin-1-ium-1-olate
(3S,4R)-4-(2-methylphenyl)-1-[2-(2-oxoazepan-1-yl)acetyl]pyrrolidine-3-carboxylic acid
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-[(2-ethylpyrimidin-4-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one