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N5,N5-dimethyl-N6-[(3-methylpyridin-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
1-[1-ethyl-5-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methyl-3-oxo-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-6-carboxamide
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}acetamide
2-{3-[({1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}carbamoyl)amino]phenyl}acetamide
3-[1-(2H-1,3-benzodioxol-5-yl)propan-2-yl]-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1,2-oxazole-5-carboxamide
2-phenyl-1-{1-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}ethan-1-ol
2-{[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-1-ethyl-1H-imidazole
2-{6-[4-(2-chlorophenyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-methylpyridine-3-carboxamide
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-(pyrrolidine-1-carbonyl)pyrazin-2-amine
3-(2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
1-[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(methylsulfanyl)ethan-1-one
7-acetamido-1-[2-(pyridin-2-yl)ethyl]-N-{[3-(trifluoromethoxy)phenyl]methyl}-1H-1,3-benzodiazole-5-carboxamide
2-{3-[2-(4-methylpentyl)morpholin-4-yl]-3-oxopropyl}-2,3-dihydro-1H-isoindol-1-one
3-[2-(propan-2-yl)-1H-imidazol-1-yl]-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-cyclopropyl-3,4-difluoro-N-({3-[2-(piperidin-1-yl)ethoxy]phenyl}methyl)benzene-1-sulfonamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(4-propylbenzoyl)pyrrolidin-3-yl]methanol
1-[5-(2-methoxy-4-methylphenoxymethyl)-1,2-oxazole-3-carbonyl]azepane
N-[(1S,2R)-2-(cyclooctylamino)cyclobutyl]-2-(1H-1,2,4-triazol-1-yl)benzamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(2-oxopyrrolidin-1-yl)ethyl]benzamide
(2R,6R)-10-methoxy-4-(3,3,4,4-tetrafluorobutyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
methyl (2S,4S)-1-methyl-4-[(morpholine-4-sulfonyl)amino]pyrrolidine-2-carboxylate
2-methyl-5-[2-(piperidin-1-ylmethyl)-1,4-oxazepane-4-carbonyl]phenol
4-{4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydrophthalazin-1-one
2-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidine
(2S,4S)-4-amino-N,N-diethyl-1-{2-[4-(methylsulfanyl)phenyl]acetyl}pyrrolidine-2-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-hydroxyphenyl)ethan-1-one
2-(2-chlorophenyl)-3-methyl-N-[3-(1H-pyrazol-1-yl)propyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-{1-oxo-1-[3-(pyridin-4-yl)azetidin-1-yl]butan-2-yl}-2,3-dihydro-1H-isoindol-1-one
2-(1H-1,3-benzodiazole-5-carbonyl)-7-{[4-(propan-2-yl)phenyl]methyl}-2,7-diazaspiro[4.5]decane
2-(4-chlorophenyl)-5-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
8-(5-ethyl-1,2,4-oxadiazol-3-yl)-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]-1-(1-methylpiperidin-4-yl)piperazin-2-yl}ethan-1-ol
2-{[(1S,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
2-[4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)amino}methyl)phenyl]-5-methyl-6-(trifluoromethyl)-3,4-dihydropyrimidin-4-one
1-{1-[2-(ethylamino)pyrimidine-5-carbonyl]piperidin-3-yl}-3-phenylpropan-1-one
(4aS,7aR)-1-(2-methyl-1,3-benzoxazole-6-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 5-[(1-ethylpiperidin-4-yl)amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-(3-methoxyphenyl)-1-(1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine
1-{2-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidin-2-one
3-(furan-2-ylmethyl)-5-propyl-5-{1-[2-(2,4,6-trifluorophenyl)acetyl]piperidin-4-yl}imidazolidine-2,4-dione
methyl 3-[2-oxo-6-(pyridin-4-ylmethoxy)-4-[2-(1,3-thiazol-4-yl)acetyl]-1,4-diazepan-1-yl]propanoate
{[1-butyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
4-[(4-{3-[benzyl(methyl)amino]-2-hydroxypropoxy}phenyl)methyl]-3,3-dimethylpiperazin-2-one
methyl 2-[3-(3-chlorophenyl)-3-(2-hydroxyphenyl)-N-methylpropanamido]acetate
3-ethyl-1-methyl-N-{[3-methyl-7-(2-methylbutanoyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1H-pyrazole-5-carboxamide
N-({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine