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4-{[(4aS,7aR)-4-(2-methylpropanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzonitrile
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methylphenyl)methyl]piperazin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-(1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}piperidin-4-yl)propanamide
[(3R,4R)-1-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(2R,3R,6R)-5-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(3,4-dimethylphenyl)methyl]piperidin-4-yl}oxy)benzamide
N-cyclopropyl-1-(1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-4-yl)-1H-1,2,3-triazole-4-carboxamide
(2S)-3-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-ylmethyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl}propane-1,2-diol
5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
N-methyl-N-{1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]-2-(2-methylphenyl)ethyl}-2-(1H-pyrazol-1-yl)acetamide
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-methoxyphenol
N,N-diethyl-1-[(1s,4s)-4-(thiophene-2-sulfonamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
1-(5-chloropyridin-2-yl)-4-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
4-(4-cyclobutanecarbonylpiperazin-1-yl)-2-(pyridin-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-(2-ethyl-1H-1,3-benzodiazol-1-yl)-N-[2-(pyridin-4-yl)ethyl]butanamide
2-methyl-5-{4-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]piperazine-1-carbonyl}phenol
3-fluoro-N,4-dimethyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
4-{[5-(1H-pyrazol-5-yl)furan-2-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(3S,4R)-1-methyl-3-({[(1-methyl-1H-pyrazol-4-yl)methyl](propan-2-yl)amino}methyl)piperidin-4-ol
1-(furan-2-ylmethyl)-N-[(3-propyl-1,2-oxazol-5-yl)methyl]piperidine-4-carboxamide
methyl 4-{[4-(morpholin-4-ylmethyl)phenyl]carbamoyl}piperazine-1-carboxylate
5-(1-tert-butyl-5-oxopyrrolidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
9-[3-(4-hydroxyphenyl)propanoyl]-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-chloro-5-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,2-dihydropyridin-2-one
3-[1-(2-cyclopentylacetyl)piperidin-4-yl]-N-cyclopropylpropanamide
N-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]amine
(1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,3-benzodiazol-2-yl)methanol
1-(oxan-3-ylmethyl)-2-(5-propylfuran-2-yl)-1H-imidazole
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(furan-2-ylmethyl)-N-(prop-2-yn-1-yl)benzamide
6-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}pyridine-2-carbonitrile
2-(4-acetyl-1,4-diazepan-1-yl)-2-[4-(methylsulfanyl)phenyl]acetic acid
2-(carbamoylamino)-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}acetamide
3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[1-(1,3-thiazol-2-yl)ethyl]benzamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)propanamide
3-(1-methyl-1H-pyrazol-5-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}propanamide
(2S)-6-amino-2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)hexanoic acid
N,N-diethyl-1-[1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperidine-3-carboxamide
1-[3-({[3-(3,4-dimethylphenyl)-1H-pyrazol-4-yl]methyl}amino)propyl]pyrrolidin-2-one
N-[2-(2,6-dimethylmorpholin-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
1-[(2-fluorophenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
4-methoxy-2-{[7-(2-methylphenyl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}phenol
2-(2-{2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-ylmethyl}phenoxy)acetic acid
2-(3-fluorophenoxymethyl)-N-[(1-hydroxycyclohexyl)methyl]-1,3-oxazole-4-carboxamide
3-(4-fluorophenyl)-N-(1H-indol-3-yl)-1H-pyrazole-5-carboxamide
N-({3-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}methyl)acetamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(1-tert-butyl-5-oxopyrrolidin-3-yl)methyl]-N-methylacetamide
5-methyl-1-[(1-methyl-1H-imidazol-2-yl)methyl]-5-(4-methylpent-3-en-1-yl)piperidin-2-one
5-methyl-N-{[4-(2-methylphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
2-{4-[(4-ethoxyphenyl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol