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N-ethyl-4-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetamido]piperidine-1-carboxamide
(1S,5R)-3-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(dimethylamino)ethyl]-3-(oxolan-2-ylmethyl)-1-[4-(1H-pyrazol-5-yl)phenyl]urea
N-(4-chloro-2-methylphenyl)-5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[(5-methylthiophen-2-yl)methyl]-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazine
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazole-5-carboxamide
2-(2-fluorophenyl)-N-{[8-(pyridin-4-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3,3-dimethyl-1-[(5-{[2-(methylsulfanyl)phenyl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]urea
5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
N-(2-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)oxolane-2-carboxamide
methyl 3-benzoyl-7-oxo-9-[3-(pyridin-4-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{3-[1-(2-methylpyridin-4-yl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}acetamide
3-(2-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}-2-oxoethyl)-5,5-dimethylimidazolidine-2,4-dione
5,8-dichloro-3-(3-hydroxy-2,2-dimethylpropyl)-3,4-dihydroquinazolin-4-one
1-[(3,4-difluorophenyl)methyl]-4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine
(3S,4R)-4-(2-methoxyphenyl)-1-(5-methyl-1,3-oxazole-4-carbonyl)pyrrolidine-3-carboxylic acid
1-{2-[1-(cyclohexylmethyl)-2,5-dioxo-3-phenylpyrrolidin-3-yl]acetyl}piperidine-4-carboxamide
(1R,5R)-6-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonane
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(2,3-dihydro-1H-inden-1-yl)acetamide
(2R)-2-amino-1-(3,3-diphenylpiperidin-1-yl)propan-1-one
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-methyl-2-oxo-1,2,5,6,7,8-hexahydroquinoline-3-carboxamide
2-(4-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-3-[2-(2-methylphenyl)ethyl]piperidine
N-[phenyl(pyridin-4-yl)methyl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
6-methoxy-4-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-1-(pyridin-3-ylmethyl)-1,4-diazepan-2-one
1-cycloheptyl-6-oxo-N-{[1-(piperidin-1-yl)cyclopentyl]methyl}piperidine-3-carboxamide
1-methyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
6-[2-(5-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetyl]-N-phenyl-6-azaspiro[2.5]octane-1-carboxamide
2-methyl-1-{2-[3-(pyridazin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1H-indole
3-[(3S,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
2-(3-methylbutyl)-8-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-4-cyclopropyl-1-(3-methylpyrazin-2-yl)pyrrolidin-3-yl]oxane-4-carboxamide
4-(hydroxymethyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-ol
N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-3-(4H-1,2,4-triazol-4-yl)benzamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethan-1-one
4-{[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]methyl}-1H-pyrazole-3-carboxylic acid
3-methyl-1-(2-methylphenyl)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}urea
N-ethyl-N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
N-(3-chloro-2-fluorophenyl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
(3S,4S)-1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
2-{4-[(6-fluoroquinolin-2-yl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3-methyl-7-{[3-(5-methylfuran-2-yl)phenyl]methyl}-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
4-phenyl-1-[(1-propyl-1H-pyrazol-4-yl)methyl]-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-imidazole
3-hydroxy-3-({methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)-1-[(3-methylphenyl)methyl]piperidin-2-one
ethyl 4-[6-(cyclohex-3-en-1-ylmethyl)-6-azaspiro[2.5]octane-1-amido]piperidine-1-carboxylate
N-({1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-3-yl}methyl)furan-2-carboxamide
{5-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
N-(1-{1-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylthiophene-3-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl](methyl)[(2-methyl-1,3-thiazol-4-yl)methyl]amine