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1-methyl-4-[1-methyl-5-(thiophen-2-yl)-1H-pyrazole-3-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{[4-(3-methylbutyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
N-[2-(2,4-difluorophenyl)-1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]ethyl]-N-methylpropanamide
N-ethyl-5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
1-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(1H-imidazol-2-yl)-N-[3-(methylamino)propyl]benzamide
ethyl 5-[(2,1,3-benzothiadiazol-5-ylmethyl)carbamoyl]-1H-imidazole-4-carboxylate
N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}imidazo[1,2-a]pyridine-6-carboxamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[4-(propan-2-yl)-1,3-thiazol-2-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
4-{5-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-3-phenyl-1H-pyrazole
9-methyl-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-9H-carbazole-3-carboxamide
4-chloro-1-methyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-1H-pyrazole-3-carboxamide
2-cyano-N-(furan-2-ylmethyl)-N-(3-methylbutan-2-yl)benzamide
2-(2-oxoazepan-1-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
N-[(3R,4S)-1-methanesulfonyl-4-(propan-2-yl)pyrrolidin-3-yl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
(3S)-1-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}pyrrolidin-3-ol
N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-2,3-dimethoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
N-[2-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-2-yl)ethyl]acetamide
4-[(3,4-dichlorophenyl)methyl]-1,4-oxazepan-5-one
2-(1H-imidazol-2-yl)-N-{2-[(trifluoromethyl)sulfanyl]ethyl}benzamide
(3aR,6aR)-2-cyclopropanecarbonyl-5-(2,2-dimethylpent-4-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(pyrrolidin-1-yl)ethan-1-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
[(3R,4R)-1-(5-chlorothiophene-2-carbonyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N-(2-methoxyethyl)-1-propyl-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-(4-acetylbenzenesulfonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1-cyclopentanecarbonylpiperidin-3-yl)-4-(4-methoxyphenyl)piperazine
3-(3-methyl-1,2,4-thiadiazol-5-yl)-1-{[1-(piperidin-1-yl)cyclohexyl]methyl}urea
ethyl 2,4-dimethyl-5-[3-(3-methylphenoxy)azetidine-1-carbonyl]-1H-pyrrole-3-carboxylate
8-[2-(4-fluorophenoxy)ethyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
4-(4-fluorophenyl)-N-{[8-(pyridin-3-ylmethyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}benzamide
2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}-N-(1-phenylethyl)acetamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-2-(methylsulfanyl)pyridine-3-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-fluoroethyl)piperidine-3-carboxamide
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-3-(5-phenyl-2H-1,2,3,4-tetrazol-2-yl)propan-1-one
4-{[2-(1H-imidazol-1-yl)ethyl]sulfamoyl}-N-[(3S)-pyrrolidin-3-yl]benzamide
N-[(5-{[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]methyl}furan-2-yl)methyl]-N-methylmethanesulfonamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(1-methyl-6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)piperidin-3-yl]propanamide
3-{1-[2-(ethanesulfonyl)acetyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-[2-(pyridin-3-yl)ethyl]acetamide
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
4-{5-[3-(propan-2-yl)-1,2-oxazol-5-yl]-1,2,4-oxadiazol-3-yl}pyridine
1-{4-[(3aS,6aS)-1-cyclopentanecarbonyl-octahydropyrrolo[2,3-c]pyrrole-5-carbonyl]-1H-pyrazol-3-yl}-1H-1,2,3,4-tetrazole
N-{4-[(2-methanesulfonylethyl)carbamoyl]phenyl}-2-methylfuran-3-carboxamide
2-methyl-1-[3-(2-methylphenoxy)azetidin-1-yl]-3-(morpholin-4-yl)propan-1-one
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(2-methylphenoxy)azetidine
N-{[5-chloro-7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}quinoline-2-carboxamide
ethyl 4-{1-[2-(1H-imidazol-1-yl)acetyl]piperidin-3-yl}piperazine-1-carboxylate
1-(2-methoxyethyl)-8-[(4-methyl-1H-imidazol-2-yl)methyl]-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}-2,3,4,5-tetrahydropyridazin-3-one