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1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-N-[2-(pyrazin-2-yl)ethyl]piperidine-4-carboxamide
3-{[1-({3-methanesulfonylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidin-4-yl]oxy}pyridine
[4-({1-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
(3S,4S)-1-(benzenesulfonyl)-4-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}pyrrolidin-3-ol
1-(5-ethyl-2-methylpyrimidin-4-yl)-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-[4-({[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
1-[3-({[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}methyl)phenoxy]-3-(4-ethylpiperazin-1-yl)propan-2-ol
6-{[3-(2-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
N3-benzyl-4-oxo-1-(propan-2-yl)-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
3-benzyl-1-(3-methoxypropyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-ethyl-N-{[7-(2-fluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-methyl-1H-pyrazole-5-carboxamide
1-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]piperidin-3-yl}pyrrolidin-2-one
(3R)-1-[(1-{1-[(1r,4r)-4-methylcyclohexanecarbonyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]pyrrolidin-3-amine
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}pyrimidin-2-amine
(2R,6R)-4-(1-ethylpiperidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(4-chlorophenyl)-4-[(4-methoxypyridin-2-yl)methyl]morpholine
N-(furan-2-ylmethyl)-9-methoxy-7-oxo-3-{[4-(trifluoromethoxy)phenyl]methyl}-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidine
4-{4-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidin-1-yl}-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-(2-butyl-1H-imidazol-4-yl)-1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-1H-imidazole
2-(2-phenyl-1H-imidazol-1-yl)-N-(3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}propyl)acetamide
1-[(3-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)methyl]-1H-pyrazole
N-methyl-N-(1-methylpiperidin-4-yl)-5-(4-phenylazepane-1-carbonyl)pyridin-2-amine
N-[2-(2,5-dimethylphenoxy)ethyl]-6-(2-hydroxyethyl)-N-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-(2-chlorophenyl)-1-(1,4-oxazepan-6-ylmethyl)urea
1-{4-[2-(2-ethylpiperidine-1-carbonyl)phenoxy]piperidin-1-yl}-2-methoxyethan-1-one
N-[2-(4-fluorophenyl)-2-(piperidin-1-yl)ethyl]-3-(methoxymethyl)benzamide
2-[4-(2,1,3-benzoxadiazol-5-ylmethyl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
2-(1-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperidin-3-yl)-4-methyl-1H-1,3-benzodiazole
3-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
4-ethyl-1-methyl-3-{[1-(2-methyloxolane-2-carbonyl)piperidin-4-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-5-ethyl-2-methylpyrimidin-4-amine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclopropanesulfonamide
2-[2-(1-methylpiperidin-2-yl)ethyl]-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
(3S,4S)-1-(5-methylpyridine-3-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-acetamido-1-ethyl-2-(3-methoxyphenyl)-N,N-bis(prop-2-en-1-yl)-1H-1,3-benzodiazole-7-carboxamide
2-(1-phenylcyclohexyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-phenyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-3-methoxypropan-1-one
7-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-benzofuran-2-carboxamide
5-[(2-chlorophenyl)methyl]-3-(cyclopropylmethyl)-5-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}imidazolidine-2,4-dione
ethyl 4-[(4-methoxyphenyl)methyl]-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)piperidine-4-carboxylate
3-(2H-1,3-benzodioxol-5-yl)-N-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-3-phenylpropanamide
1-{[(3R,4R)-4-(hydroxymethyl)-1-(5-methylthiophene-2-carbonyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[2-(morpholin-4-yl)-2-(pyridin-4-yl)ethyl]pyrrolidin-2-one
N-[(2-methoxyphenyl)methyl]-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
2-(4-fluorophenyl)-4-(5-propyl-1,3,4-oxadiazol-2-yl)morpholine