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N-{1-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-1H-pyrazol-4-yl}thiophene-3-carboxamide
1-[2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
N-benzyl-3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
2-{[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
N-benzyl-3-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}benzamide
2-methanesulfonyl-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
9-methoxy-N-methyl-3-[2-(4-methylphenoxy)acetyl]-7-oxo-N-(thiophen-3-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
N-ethyl-2-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyrimidin-4-amine
N-[2-(4-fluorobenzenesulfonyl)ethyl]oxolane-3-carboxamide
2-[1-(4-methoxyphenyl)cyclopentanecarbonyl]-2,7-diazaspiro[4.5]decan-6-one
6-(2-aminoethyl)-N,2-dimethyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidin-4-amine
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
2-(2-{1-[1-(2-phenylethyl)-1H-1,2,3-triazole-4-carbonyl]piperidin-2-yl}ethyl)pyridine
3-({[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}carbamoyl)pyridin-1-ium-1-olate
2-(2-hydroxyphenyl)-N-methyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
4-ethyl-1-[(4-fluorophenyl)methyl]-1,4-diazepan-5-one
4-[(3-fluorophenyl)methyl]-3-{2-[4-(3-methoxypropyl)piperidin-1-yl]-2-oxoethyl}piperazin-2-one
1-(2-methoxy-5-{[(1-propylpiperidin-4-yl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
3-cyclopentyl-1-ethyl-5-{7-methylpyrazolo[1,5-a]pyrimidin-6-yl}-1H-1,2,4-triazole
N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
3-chloro-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]thiophene-2-carboxamide
2-[4-(2-chloro-6-methoxyphenyl)phenyl]-N-methylacetamide
2-{[1-(1-methyl-1H-pyrazol-5-yl)propyl]amino}propane-1,3-diol
2-[1-(propan-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
N,N,5-trimethyl-2-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyrimidin-4-amine
N-[(4-methoxyphenyl)methyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
(3S,4S)-N-[2-(2-ethoxyethoxy)phenyl]-3,4-bis(hydroxymethyl)pyrrolidine-1-carboxamide
N,4-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-5-methyl-1-(3-methylphenyl)piperazin-2-one
N-{1-[1-(5-acetylthiophene-2-carbonyl)piperidin-4-yl]-2-(2,4-difluorophenyl)ethyl}-N-methylcyclopropanecarboxamide
1-[3-(furan-2-yl)-3-phenylpropyl]-3-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)urea
1-(2-methylphenyl)-4-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}piperazin-2-one
2-(4-{[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1-methylpiperazin-2-yl)ethan-1-ol
(4aS,7aR)-1-[(1R,5S,6R)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-chloro-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-4-fluorobenzamide
4-{4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}quinoline
N-cyclohexyl-6-(2-hydroxyethyl)-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[2-(2-methylphenyl)ethyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperidine-3-carboxamide
1-[2-(4-chlorophenyl)ethyl]-5-(pyrrolidine-1-carbonyl)piperidin-2-one
N-(4-ethylphenyl)-3-[2-(furan-3-yl)-1H-imidazol-1-yl]propanamide
N-{[5-(3-cyclopentylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
4-[(2S)-4-methyl-2-phenylpiperazine-1-carbonyl]-2-(1H-pyrazol-4-yl)quinoline
N-ethyl-N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-2-phenylethyl)oxane-4-carboxamide
(1S,5R)-6-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(3R,4R)-1-(2,6-dimethylquinoline-4-carbonyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
methyl 2-{3-[({1-[(3-methoxyphenyl)methyl]piperidin-3-yl}amino)methyl]-1H-indol-1-yl}acetate
1-(1H-indazol-7-yl)-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one