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N-(furan-2-ylmethyl)-1-{2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}piperidine-4-carboxamide
2-(2-chloro-4-fluorophenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}acetamide
4-cyclopropyl-6-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]pyrimidine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[1-(1-methyl-1H-pyrazol-5-yl)propyl]amine
1-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-3-yl]-4-[3-(trifluoromethyl)phenyl]piperazine
{[3-(3-fluoro-4-methoxyphenyl)-1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl})(propan-2-yl)amine
1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidin-3-amine
N-[2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-4-methylbenzamide
N-[cyclopropyl(pyridin-2-yl)methyl]-N,2,8-trimethylquinoline-4-carboxamide
4-(2-ethylbutanoyl)-1-(4-methoxyphenyl)piperazin-2-one
4-(1H-indol-3-yl)-N-(5-oxo-1-phenylpyrrolidin-3-yl)butanamide
(1s,4s)-4-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}cyclohexan-1-ol
2-{[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
{2-[1-(3,5-dimethylphenyl)-1H-1,2,4-triazol-5-yl]ethyl}dimethylamine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(3,4-dimethoxyphenyl)methyl]-N5-[2-(1-methylpyrrolidin-2-yl)ethyl]piperidine-3,5-dicarboxamide
1-(2-methoxy-5-{[(1-phenylpiperidin-4-yl)amino]methyl}phenoxy)-3-(pyrrolidin-1-yl)propan-2-ol
N-(2-{7-[(2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
N-{[5-fluoro-7-(pyridin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-phenoxypropanamide
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl){[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
3-{4-[(2-ethyl-4-methyl-3-oxopiperazin-1-yl)methyl]-1H-pyrazol-1-yl}propanoic acid
2-methyl-4-[5-(oxan-4-yl)-3-(2-phenylethyl)-1H-1,2,4-triazol-1-yl]pyridine
4-(2-methoxyphenyl)-3-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazole
5-[1-(2-cyclopentylacetyl)piperidin-4-yl]-5-(3-methylbutyl)-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-amino-4-phenyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl}pyrimidine-5-carboxamide
2-[4-({3-[5-phenyl-2-(pyridin-4-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]benzamide
(2E)-3-(furan-2-yl)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]prop-2-en-1-one
1-(5-fluoropyridine-3-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
1-[(4aR,8aR)-7-(5-ethyl-1,3,4-oxadiazol-2-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
4-phenyl-N-{[1-(pyrrolidine-1-carbonyl)piperidin-3-yl]methyl}benzamide
{3-[(2-fluorophenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
2-amino-N-[(3R,4S)-4-(propan-2-yl)-1-[5-(propan-2-yl)pyrimidin-4-yl]pyrrolidin-3-yl]acetamide
5-(dimethylamino)-2-(2-propoxyethyl)-2,3-dihydropyridazin-3-one
{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}({[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl})(pyridin-4-ylmethyl)amine
2-[(1S,5R)-3-[(4-ethoxyphenyl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
2-methyl-6-{1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}pyrimidin-4-ol
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-(1-propyl-1H-pyrazole-5-carbonyl)-1,4-diazepane
6-{2-amino-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-5-yl}-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
methyl 2-(2-{[2-(2H-1,3-benzodioxol-5-yl)acetamido]methyl}-5-methyl-2,3-dihydro-1-benzofuran-7-yl)benzoate
3-ethyl-4-({4-[(4-fluoro-3-methoxyphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperazin-2-one
6-[7-(oxan-4-yl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]pyridine-2-carboxylic acid
1-(2-methoxyphenyl)-4-[(5-propyl-1,3,4-oxadiazol-2-yl)amino]pyrrolidin-2-one
(2S,4R)-4-amino-N-methyl-1-{4-[(pyridin-2-ylsulfanyl)methyl]benzoyl}pyrrolidine-2-carboxamide
5-[benzyl(methyl)amino]-2-[(2-methyl-1,3-oxazol-4-yl)methyl]-2,3-dihydropyridazin-3-one
1-(5-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-pyrazol-3-yl)ethan-1-one
1-methyl-N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)-1H-pyrazole-4-carboxamide
[5-({[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]amino}methyl)furan-2-yl]methanol
N-{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}-2-(2-methoxyethyl)-1,3-benzoxazole-6-carboxamide
2-[4-(dimethyl-1,3-thiazole-5-carbonyl)morpholin-3-yl]-N-(pyridin-3-ylmethyl)acetamide