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(2E)-N-{[7-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-phenylprop-2-enamide
3-ethyl-N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-1-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-5-carboxamide
N-(cyclopropylmethyl)-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-(oxolan-2-ylmethyl)acetamide
3-(methoxymethyl)-1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-cyclohexyl-1-methyl-N-(pyridin-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-({4-[2-(4-ethylpiperazin-1-yl)ethoxy]phenyl}methyl)-2-methyl-1,4-oxazepane
3-(2H-1,3-benzodioxol-5-ylmethyl)-5-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-5-ethylimidazolidine-2,4-dione
(3aR,6aR)-2-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(3-methyl-1H-pyrazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(4aR,7aS)-1-acetyl-4-(3-hydroxybenzoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[1-(2-amino-6-methylpyrimidine-4-carbonyl)piperidin-3-yl]methyl}-4-phenylbenzamide
3-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyridine
3-methyl-2-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}pyridine
4-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
5-(2,3-dihydro-1,4-benzodioxin-6-yl)-N-(prop-2-en-1-yl)furan-2-carboxamide
(3S,4R)-1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
N-(1-{7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-3-methylbutyl)acetamide
N-{[7-chloro-5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopent-1-ene-1-carboxamide
3-[(2,5-dimethylphenyl)methyl]-9-methoxy-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-(2-methoxyethoxy)-1-(1H-pyrazole-4-carbonyl)piperidine
1-[(1r,4r)-4-hydroxycyclohexyl]-3-[3-(1,3-thiazol-4-yl)phenyl]urea
1-[(4-methoxyphenyl)methyl]-3-(pyridin-4-yl)-6-(quinolin-4-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
5-(1,2-oxazinane-2-carbonyl)-1-(2-phenylethyl)piperidin-2-one
2-{2-[2-(dimethylamino)ethyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-2-oxo-N-phenylacetamide
1-(6-{3-[(2-fluorophenyl)methyl]-3-(hydroxymethyl)piperidin-1-yl}pyridin-3-yl)ethan-1-one
N-(1-{7-[(2-hydroxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
2-(2-{[4-(pyridin-3-yl)piperazin-1-yl]methyl}phenoxy)propanoic acid
2-[(3,3-dimethylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
methyl 5-cyano-2-methyl-6-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyridine-3-carboxylate
N-[2-(3,5-dimethylphenoxy)ethyl]-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methylacetamide
1-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-4-(2-methoxyphenyl)piperazine
4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
N-[2-(2-fluorophenyl)-2-hydroxyethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
1-{5-cyclopropyl-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}-N,N-diethylpyrrolidin-3-amine
N-[(2-chloropyridin-3-yl)methyl]-N,3,5-trimethyl-1,2-oxazole-4-carboxamide
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-ethyl-N-[(5-methylfuran-2-yl)methyl]acetamide
3-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]-5,6-dihydro-1,4-dioxine-2-carboxamide
N-[2-methyl-2-(morpholin-4-yl)propyl]-1-propyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(ethanesulfonyl)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]piperidine-3-carboxamide
7-(propan-2-yl)-2-[2-(pyrimidin-2-ylsulfanyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N,N-dimethyl-5-{[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}pyridin-2-amine
2,2-dimethyl-4-oxo-N-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-3,4-dihydro-2H-pyran-6-carboxamide
N-(furan-2-ylmethyl)-2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-propylacetamide
4-(furan-2-ylmethyl)-3-[2-(2-hydroxyphenyl)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-cyclopentyl-4-{4-methoxy-2-[3-(methoxymethyl)pyrrolidine-1-carbonyl]phenoxy}piperidine
1-{pyrazolo[1,5-a]pyridine-3-carbonyl}-2-[2-(thiophen-2-yl)ethyl]piperidine
N-[(3,4-dimethoxyphenyl)methyl]-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(pyridin-2-ylmethyl)acetamide
5-[(2,4-dimethoxy-3-methylphenyl)methyl]-N,N-dimethyl-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-cyclopropyl-3-(2-fluorophenyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-5-carboxamide