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(1S,6R)-3-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonane
1-(5-methanesulfonyl-2-methylphenyl)-3-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[1-(thiophen-2-yl)propan-2-yl]benzamide
1-{3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-phenylpropan-1-one
5,6-dimethyl-2-oxo-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]-1,2-dihydropyridine-3-carboxamide
N,1-bis(propan-2-yl)-2-[5-(1H-pyrazol-3-yl)furan-2-yl]-1H-1,3-benzodiazole-5-sulfonamide
2-methoxy-N,4-dimethyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1,3-thiazole-5-carboxamide
N-(1H-1,3-benzodiazol-2-ylmethyl)-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
methyl (1R,3S,3aR,6aS)-5-benzyl-1-methyl-3-(1-methyl-1H-imidazol-5-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-methyl-2-(3-oxo-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}piperazin-2-yl)acetamide
1-methyl-4-({4-methyl-5-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)piperazine
1-(7-methoxy-4-methylquinazolin-2-yl)-N-methyl-N-[(4-methylphenyl)methyl]piperidine-4-carboxamide
N,N-dimethyl-5-{[methyl({[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl})amino]methyl}pyridin-2-amine
N-{3-[cyclopentyl(methyl)amino]propyl}-6-ethylpyrimidin-4-amine
N-(1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-2-(2-fluorophenyl)ethyl)-N,2-dimethylfuran-3-carboxamide
2-(3-methoxyphenyl)-N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,3-benzoxazole-6-carboxamide
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylacetamide
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)naphthalene-1-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-3-{octahydropyrrolo[1,2-a]piperazine-2-carbonyl}-1,2-oxazole
2,6-dimethyl-N-[2-(6-oxo-3-phenyl-1,6-dihydropyridazin-1-yl)ethyl]pyrimidine-4-carboxamide
2-[(4-fluorophenyl)methyl]-4-{[1-(pyridin-4-yl)-1H-pyrrol-2-yl]methyl}morpholine
4-(piperidin-1-yl)-1-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine
2-({4-[2-amino-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperazin-1-yl}methyl)-6-methylpyridin-3-ol
1-{[5-methoxy-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(1H-pyrazol-1-ylmethyl)piperidine
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[3-(piperidin-1-yl)propyl]benzamide
N-[1-(1-{[1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]oxolane-3-carboxamide
2-[4-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)piperazin-1-yl]-N-(propan-2-yl)acetamide
8-chloro-N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}quinoline-2-carboxamide
3-(3,4-difluorophenyl)-N-[(3-methyloxetan-3-yl)methyl]propanamide
(3S,4S)-4-cyclopropyl-1-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]pyrrolidine-3-carboxylic acid
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-(naphthalene-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(2,1,3-benzothiadiazol-5-ylmethyl)({[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)furan-2-carboxamide
5-ethyl-2-{[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
2-(4-methoxy-2-methylphenyl)-3-(pyrrolidin-1-yl)pyrazine
{3-[(3-chlorophenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methanol
2-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-6-methylpyridine-3-carboxamide
2-(2-{[3-(hydroxymethyl)morpholin-4-yl]methyl}-4-(pyrimidin-2-yl)phenoxy)acetic acid
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(pyridin-2-yl)acetamide
1-[(5-methylthiophen-2-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
ethyl 4-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]piperazine-1-carboxylate
6-(2,5-dimethylfuran-3-yl)-N,N-bis(2-hydroxyethyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-[(4-methoxyphenyl)methyl]pyridin-2-amine
N-[2-(7-{[4-(propan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)ethyl]cyclohexanecarboxamide
[4-({[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)amino}methyl)oxan-4-yl]methanol
1-(6-cyanopyridin-2-yl)-N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]piperidine-4-carboxamide
N-cyclobutyl-4-{[3-(methylsulfanyl)propyl]sulfamoyl}benzamide
6-cyclopentyl-2-methoxy-3-{[(5-methoxypyrimidin-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-[3-(trifluoromethyl)phenyl]piperidin-4-ol
7-(cyclohexylmethyl)-2-(5-methyl-1,2-oxazole-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one