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1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-3-[4-(dimethylamino)phenyl]propan-1-one
2-[(dimethylamino)methyl]-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-1,3-thiazole-4-carboxamide
2-[1-(3,5-dichloro-4-methylbenzoyl)pyrrolidin-2-yl]ethan-1-ol
2-(2,4-dichlorophenoxy)-N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]acetamide
4-{[5-(1-cyclohexanecarbonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
3-(dimethyl-1,2-oxazol-4-yl)-1-(4-phenyl-1,4-diazepan-1-yl)propan-1-one
N-ethyl-N-[2-(3-methylphenoxy)ethyl]but-3-enamide
9-methyl-3-(2-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-3,9-diazaspiro[5.6]dodecane
ethyl 4-(7-fluoro-3-methyl-1-benzofuran-2-amido)piperidine-1-carboxylate
2-({3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]phenyl}amino)acetic acid
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-2-phenylethyl)methylamine
1-methyl-4-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]imidazolidin-2-one
2-fluoro-N-[1-(pyridin-2-ylmethyl)azepan-3-yl]benzene-1-sulfonamide
[2-(4-methoxyphenyl)ethyl][(1-methylpiperidin-4-yl)methyl]{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-4-(pyrimidin-2-yl)-1,4-diazepane
2-methyl-N-[(5-oxopyrrolidin-2-yl)methyl]-1-benzofuran-7-carboxamide
[2-(7-{[(5-methylfuran-2-yl)methyl]sulfamoyl}-1,2,3,4-tetrahydroisoquinolin-2-yl)-2-oxoethyl]urea
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(pyrazin-2-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
methyl 2-({1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]piperidin-3-yl}formamido)acetate
2-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]benzonitrile
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-4-(piperidin-1-yl)-N-(pyridin-2-ylmethyl)benzamide
2-(dimethylamino)-1-(9-hydroxy-7-{8-thiatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[2,1-b][1,3]thiazol-6-ylmethyl})amine
6-chloro-N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-{2-[2-(pyridin-2-yl)ethyl]phenyl}propanamide
5-{8-benzyl-2,8-diazaspiro[5.5]undecane-2-carbonyl}-3,4-dihydropyrimidin-4-one
N-[(5-methylfuran-2-yl)methyl]-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
5-(3-methoxyphenoxymethyl)-N-(2-phenylpropyl)-1,2-oxazole-3-carboxamide
4-phenyl-5-[3-(1H-pyrazol-1-yl)phenyl]-1-(pyrrolidin-3-yl)-1H-imidazole
1,3-dimethyl-4-{[2-(propylamino)pyrimidin-5-yl]methyl}piperazin-2-one
1-(pyridin-3-ylmethyl)-4-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-1,4-diazepane
2-ethyl-N-[(1S,2R)-2-[(propan-2-yl)amino]cyclobutyl]pyrimidine-5-carboxamide
methyl({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})[2-(2-methylpiperidin-1-yl)ethyl]amine
N-methyl-N-(1-{1-[2-(methylsulfanyl)pyridine-3-carbonyl]piperidin-4-yl}-2-phenylethyl)thiophene-3-carboxamide
3-{1-[1-(2-ethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-1-ol
8-(1-benzofuran-2-ylmethyl)-1-methoxy-1,8-diazaspiro[4.5]decan-2-one
2-{8-benzyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}-N-ethyl-N-methylacetamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylpyridin-4-yl)-1,4-diazepane
2-{[2-(1-phenylethyl)-1H-imidazol-1-yl]methyl}pyridine
1-{[1-(4-fluorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1H-1,2,3,4-tetrazol-5-amine
1-(4-chloro-2-fluorobenzoyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
5-{3-[4-(2-ethoxyphenyl)piperazin-1-yl]-3-oxopropyl}-5-[(2-fluoro-4-methoxyphenyl)methyl]pyrrolidin-2-one
1-(cyclohexylmethyl)-3-hydroxy-3-({[(5-methylthiophen-2-yl)methyl]amino}methyl)piperidin-2-one
1-[(4aR,8aS)-1-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-decahydro-1,6-naphthyridin-6-yl]-2-phenylethan-1-one
(4aS,8aR)-1-(4-hydroxybutyl)-N,N-dimethyl-2-oxo-decahydro-1,6-naphthyridine-6-sulfonamide
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
3-{[1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-yl]methyl}benzamide
{2-[3-ethyl-4-(propan-2-yl)piperazin-1-yl]quinolin-3-yl}methanol
3-{1-[(4-cyanophenyl)methyl]piperidin-3-yl}propanamide
N-methyl-N-(quinolin-5-ylmethyl)-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide