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1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
1'-(4-fluoro-3-methylbenzoyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
methyl 3-(ethanesulfonamidomethyl)-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
6-(1,4-diazepan-1-yl)-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
1,5-dimethyl-4-{[2-(4-methylpentyl)morpholin-4-yl]methyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
4-(2H-1,3-benzodioxol-4-ylmethyl)-6-methyl-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
(5S,9aS,9bS)-5-(5-acetylthiophen-3-yl)-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
(4aR,7aS)-1-benzyl-4-(3-phenylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2R,6R)-4-{4-[(2-hydroxyethyl)sulfanyl]benzoyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-{[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,3-dimethyl-1H-1,2,4-triazole
{[(1R,5S,6S)-3-(3,5-dichloro-4-methylbenzoyl)-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
1-[(3-benzyl-1H-1,2,4-triazol-5-yl)methyl]-2-cyclopropyl-1H-1,3-benzodiazole
N-[(5-chlorothiophen-2-yl)methyl]-6-oxo-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1,3-dimethyl-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-methyl-3-phenyl-1-(pyrrolidine-1-sulfonyl)piperidine
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(methylsulfanyl)ethan-1-one
3-ethyl-5-[(2S)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}propan-1-one
6-(4-methoxyphenyl)-9-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carbonyl]-6,9-diazaspiro[4.5]decan-7-one
N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
1-phenyl-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
1-[3-(phenylamino)piperidin-1-yl]-2-(pyridin-2-ylsulfanyl)ethan-1-one
N-(4-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}phenyl)acetamide
N-[(4-methoxyphenyl)methyl]-2,4-dimethyl-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
methyl 5-(cycloheptylamino)-1-ethyl-3-(oxolane-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
4-(6-methoxypyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 3-({[1-(4-chlorophenyl)cyclobutyl]formamido}methyl)-5-[2-(thiophen-3-yl)acetamido]benzoate
2-(methylsulfanyl)-1-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}ethan-1-one
3-{1-[(1-ethyl-1H-indol-3-yl)methyl]piperidin-3-yl}-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
3-(dimethylsulfamoyl)-N-[3-(1H-imidazol-1-yl)propyl]-5-[(2-methylpropyl)amino]benzamide
2-{[3-(methanesulfonylmethyl)piperidin-1-yl]methyl}-6-methylpyridine
3-({9-methyl-3,9-diazaspiro[5.6]dodecan-3-yl}sulfonyl)benzoic acid
2,6-dimethyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]pyrimidine-4-carboxamide
3-(1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)propan-1-ol
1-{4-[3-(6-methoxynaphthalene-2-carbonyl)piperidine-1-carbonyl]thiophen-2-yl}ethan-1-one
(3S,4R)-N,N-dimethyl-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]-4-(4-methylphenyl)pyrrolidin-3-amine
2-[4-({[(5-methylpyrazin-2-yl)methyl]amino}methyl)phenoxy]-1-(morpholin-4-yl)ethan-1-one
6-amino-N-[(2,3-dimethyl-1H-indol-5-yl)methyl]pyridine-3-carboxamide
2-amino-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}ethan-1-one
1-(3-{[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
N-[2-(4-{[4-(4-fluorophenyl)-4-oxobutanamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]oxolane-2-carboxamide
N-benzyl-3,5-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1,2-oxazole-4-carboxamide
4-(4-chlorophenoxy)-1-{[2-(2,3-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
N-(1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-(4-methylpiperazin-1-yl)propanamide
N-(1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methoxybenzamide
N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-propanoylpiperidine-3-carboxamide
2-{1-[2-(3-fluorophenoxymethyl)-1,3-oxazol-4-yl]-N-methylformamido}-N-methylacetamide
2-methyl-7-[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]-2,7-diazaspiro[4.5]decane