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4-[(4-chlorophenyl)methyl]-4-(hydroxymethyl)-N-(2-methoxy-5-methylphenyl)piperidine-1-carboxamide
1-[(4-methoxyphenyl)methyl]-5-(oxolane-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
7-fluoro-3-({5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}methyl)-1,2-dihydroquinolin-2-one
N-{1-[1-(5-fluoro-1H-indole-2-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-3-ethylpiperidin-3-ol
3-({3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)phenol
2-amino-4-(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)-6-cyclopropanecarbonyl-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
(1-{[(5-cyclobutyl-1,3,4-oxadiazol-2-yl)(methyl)amino]methyl}cyclopentyl)methanol
2-(4-fluorophenyl)-N-[2-(1H-imidazol-4-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
5-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]-4-methyl-1,2,3-thiadiazole
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
5-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline
1-[1-(cyclohexylmethyl)-1H-1,2,3-triazole-4-carbonyl]-4-[3-(trifluoromethyl)phenyl]piperazine
(4aS,8aR)-2-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-decahydroisoquinoline
N-[2-(dimethylamino)ethyl]-5-(1-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[1-(quinolin-5-ylmethyl)pyrrolidin-3-yl]benzoic acid
7-(cyclopropylmethyl)-2-[4-(2-methylpropyl)benzoyl]-2,7-diazaspiro[4.5]decan-6-one
N-(propan-2-yl)-2-(3-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}-1H-indol-1-yl)acetamide
8-fluoro-2-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]quinoline
N-cyclopentyl-3-[(3R)-3-hydroxy-3,4,4-trimethylpyrrolidin-1-yl]propanamide
(4aR,8aS)-1-(2-cyclohexylethyl)-6-[4-(1H-imidazol-1-yl)benzoyl]-decahydro-1,6-naphthyridin-2-one
1-(3-chlorothiophene-2-carbonyl)-3-[4-(3,4-difluorophenyl)-1H-pyrazol-5-yl]piperidine
{5-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(furan-2-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}methanol
3-(2-methoxybenzoyl)-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
1-(oxolan-2-ylmethyl)-4-phenylazepane
4-[(2S)-2-amino-2-[3-(furan-2-yl)-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl]phenol
3-(3,4-dimethylphenyl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-(2-phenylethyl)propanamide
methyl[(2E)-2-methyl-3-phenylprop-2-en-1-yl][1-(pyridin-2-yl)ethyl]amine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]azepan-4-amine
{2-[3-(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-2-oxoethyl}urea
5-methyl-1-{3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]pyrrolidin-1-yl}hexan-1-one
N-[1-(1-{[2-(furan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2,2-dimethylpropanamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[(5-methylthiophen-2-yl)methyl]cyclopropanamine
3-[(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)amino]-1-(3-methylpiperidin-1-yl)propan-1-one
N-{[7-(4-cyclopropanecarbonylphenyl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,4-dimethoxyphenyl)acetamide
5-(2-cyclopentylacetamido)-1-methyl-N-(3-methylbutyl)-2-(oxolan-2-yl)-1H-1,3-benzodiazole-7-carboxamide
1-[2-methyl-4-(2-methylphenyl)piperazin-1-yl]-3-(pyridin-3-yl)propan-1-one
8-[3-(4-fluorophenoxy)propyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
methyl 1-({4-[4-(morpholin-4-yl)benzoyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-4-carboxylate
2-[(1S,5R)-6-[2-(3-chlorophenoxy)acetyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]-N,N-dimethylacetamide
1-(cyclopropylmethyl)-6-(2,3-difluorobenzoyl)-3-(2-methylquinolin-5-yl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1'-[2-(benzyloxy)ethyl]-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-[(4-{5-[3-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-1-yl)sulfonyl]quinoline
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
1-(2-methoxy-4-{[methyl(2-phenoxyethyl)amino]methyl}phenoxy)-3-[methyl(propan-2-yl)amino]propan-2-ol
(3S,4S)-1-{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}-4-(dimethylamino)pyrrolidin-3-ol
3-fluoro-4-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N,N-bis(furan-2-ylmethyl)-2-(1H-imidazol-2-yl)benzamide
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(pyridin-3-yl)propyl]acetamide