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ethyl 5-{[methyl(1,2-oxazol-3-ylmethyl)amino]methyl}-1-(4-phenyl-1,3-thiazol-2-yl)-1H-pyrazole-4-carboxylate
1-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-3-methoxypiperidine
4-[2-(1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]morpholine
4-(2-{[4-(trifluoromethyl)pyrimidin-2-yl]oxy}hex-5-en-1-yl)-1,4-oxazepane
4-{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-3-ethylpiperazin-2-one
2-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
methyl 2-({1-[4-(2,4-dimethylbenzamido)phenyl]piperidin-4-yl}amino)acetate
8-(4-methylpyridin-2-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-butyl-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazole
1-[2-methoxy-5-({methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
(4aS,7aR)-N,N-dimethyl-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-sulfonamide
{3-[(3-chlorophenyl)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-3-yl}methanol
8-(3-methoxypropanoyl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-4-yl]acetamide
1-[(2-methoxypyridin-3-yl)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-methoxy-N-(2-methoxyethyl)-2-{[1-(4,4,4-trifluorobutyl)piperidin-4-yl]oxy}benzamide
N-{[1-(morpholin-4-yl)cyclohexyl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-(2-methyl-1H-imidazol-1-yl)-1-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]ethan-1-one
N-methyl-N-[(5-{6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}furan-2-yl)methyl]methanesulfonamide
1-[2-(3,4-dichlorophenyl)morpholin-4-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
6-(2-methoxyphenyl)-N-[3-(4-methoxyphenyl)propyl]pyridine-3-carboxamide
1-(7,7-dimethyl-5-{[(1-methyl-1H-pyrazol-4-yl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
2-(1H-imidazol-1-yl)-1-[7-(3-phenylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]ethan-1-one
4-(1H-imidazol-1-ylmethyl)-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
5-{2-[2-(3,4-dichlorophenyl)morpholin-4-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-amino-6-[4-(piperidin-1-yl)phenyl]-4-(pyridin-3-yl)pyridine-3-carbonitrile
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[5-(oxolan-2-yl)thiophen-2-yl]methyl}piperidine
4-benzyl-3-ethyl-1-(2-methoxy-4-methylbenzoyl)-1,4-diazepan-5-one
4-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2-(2-phenylethyl)morpholine
(2R,3S,6R)-5-(4-chloro-2-fluorobenzoyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[(1R,3R)-3-aminocyclopentyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-[3-(1H-imidazol-1-yl)propyl]-9-methoxy-3-[(3-methylphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
4-{[1-(2-hydroxyacetyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
{1-[2-({2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]piperidin-2-yl}methanol
2-(1-methyl-1H-indazol-5-yl)benzamide
1-[(4-fluorophenyl)methyl]-5-[(methylsulfanyl)methyl]-1H-1,2,4-triazole
ethyl 1-(2-hydroxyethyl)-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-(4-{1-[(2,3-dimethoxyphenyl)methyl]-1H-imidazol-2-yl}-1H-1,2,3-triazol-1-yl)piperidine
(4aS,7aR)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}acetamide
N-cycloheptyl-3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carboxamide
4-(azocan-1-yl)-N-(3-hydroxy-2,2-dimethylpropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-methyl-1,4-diazepan-5-one
1-(1,4-dithiepan-6-yl)-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-[2-(dimethylamino)ethyl]-4-ethyl-3-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[2-(cyclohexylsulfanyl)ethyl]-1-(furan-2-ylmethyl)piperidine-4-carboxamide
ethyl 4-[1-(2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}acetyl)piperidin-3-yl]piperazine-1-carboxylate
(5S,9aS,9bS)-5-(2,6-difluorophenyl)-2-[(3-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
3-{[2-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione
6-{[methyl(1H-pyrazol-3-ylmethyl)amino]methyl}naphthalen-2-ol