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N-(2H-1,3-benzodioxol-5-yl)-6-(2,2-dimethyl-4-oxo-3,4-dihydro-2H-pyran-6-carbonyl)-6-azaspiro[2.5]octane-1-carboxamide
6-(1-benzothiophen-2-yl)-N-(2,2-dimethyloxan-4-yl)-2-(morpholin-4-yl)pyridine-3-carboxamide
9-[4-(methylamino)pyrimidin-2-yl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
8-(1,3-benzothiazol-2-ylmethyl)-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
4-{3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-4-oxo-N-[2-(propan-2-yl)phenyl]butanamide
methyl 3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-3-yl]propanoate
5-{1-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}-2-(methylsulfanyl)pyrimidine
N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
6-{[3-(hydroxymethyl)-4-methylpiperazin-1-yl]methyl}pyridine-2-carboxylic acid
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-propylpiperidin-4-ol
2-[4-(1-benzothiophen-3-yl)-2-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy]-N-(3-methoxypropyl)acetamide
3-[(3R,4S)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1-[(3-methoxyphenyl)methyl]piperazin-2-one
N-({1-[3-(1,2-oxazolidin-2-yl)propanoyl]piperidin-3-yl}methyl)-4-phenylbenzamide
4-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-3-yl}-2-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}pyrimidine
N-methyl-N-(oxan-2-ylmethyl)-2-(propan-2-ylsulfanyl)acetamide
3-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-ol
(4aS,8aR)-6-(4-fluoro-3-methoxybenzoyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
3-{1-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-4-phenyl-1H-imidazol-5-yl}pyridine
N-[2-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
3-{[1-(2,3-dimethoxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
N-(1H-imidazol-2-ylmethyl)-5-(2-methoxyphenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
3-cyclopentyl-5-[(3-methoxyphenyl)methyl]-5-[1-(1,3-thiazol-2-ylmethyl)piperidin-4-yl]imidazolidine-2,4-dione
1-(2H-1,3-benzodioxol-5-ylmethyl)-N-[3-(1H-imidazol-1-yl)propyl]-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
(2E)-N-{[7-(3,6-dimethylpyrazin-2-yl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-fluorophenyl)prop-2-enamide
1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-N-(2-methoxyethyl)-5-(thiophen-2-yl)-1H-pyrazole-4-carboxamide
2-{4-[(3,3-diphenylpiperidin-1-yl)methyl]-3-methyl-1H-pyrazol-1-yl}ethan-1-ol
N-cyclopropyl-3-(1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-3-yl)propanamide
N-[3-(1,3-oxazol-5-yl)phenyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-methylacetamide
(3R,5R)-N-[2-(dimethylamino)ethyl]-1-(2-phenylethyl)-5-(pyrrolidin-1-ylmethyl)piperidine-3-carboxamide
2-methyl-4-phenyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperazine
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-(quinolin-2-ylmethyl)piperidin-3-ol
[(3R,4R)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
4-(5-chloro-2-methoxyphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
methyl 6-[(2,4-difluorophenyl)methyl]-2-[methyl(2-methylpropyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
1-[(4-hydroxy-3-methoxyphenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-1,4-diazepan-5-one
1-{3-[5-(4-hydroxyphenyl)-4-phenyl-1H-imidazol-1-yl]propyl}pyrrolidin-2-one
(3aS,6aS)-1-(2-phenylmethanesulfonylbenzoyl)-octahydropyrrolo[2,3-c]pyrrole
2-[1-(2-methoxypyridine-4-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N-[2-(adamantan-1-yl)ethyl]-2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
5-(2,6-difluorophenoxymethyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,2-oxazole-3-carboxamide
4-(1-benzofuran-2-ylmethyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
N-benzyl-5-[4-(2-fluorophenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
5-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid