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5-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N-cyclopropyl-1-[2-(phenylamino)pyrimidine-5-carbonyl]piperazine-2-carboxamide
4-[(4-fluorophenyl)methyl]-1-(2-methylfuran-3-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-{[2-(difluoromethoxy)phenyl]methyl}-4-[2-(piperidine-1-carbonyl)phenoxy]piperidine
2-(1,4-dimethylpiperazin-2-yl)-1-[4-(pyrimidin-2-yloxy)piperidin-1-yl]ethan-1-one
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-2-(pyrrolidin-1-yl)butan-1-one
N-[1-(7-{[2-(furan-2-yl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-2-methylpropyl]methanesulfonamide
4-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-3-yl)pyrimidine
4-(5-methoxyfuran-2-carbonyl)-1-(4-methoxyphenyl)-6,6-dimethylpiperazin-2-one
(2E)-3-(3-fluorophenyl)-N-[2-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)propyl]prop-2-enamide
1-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
3-(4-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}piperazin-1-yl)propanamide
1-[(1R,5R)-6-[(8-methoxyquinolin-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(2S,3R)-2-({2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazol-4-yl}formamido)-3-hydroxybutanamide
(2,3-dihydro-1-benzofuran-2-ylmethyl)({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
2-[4-(hydroxymethyl)phenyl]-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]ethan-1-one
1-cyclopentyl-4-{3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]propanoyl}piperazin-2-one
(3S,4S)-1-(6-ethyl-2-methylquinoline-4-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
2-phenyl-1-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}pyrrolidine
5-(3,4-dihydro-2H-1-benzopyran-3-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-[(4-methoxyphenyl)methyl]-6-(3-methylpiperidine-1-carbonyl)-1,3-benzoxazole
3-{2-[2-(4-fluorophenyl)morpholin-4-yl]-2-oxoethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(1-benzylpiperidin-4-yl)-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-({[(5-{[(3-fluorophenyl)methyl]sulfanyl}-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl)methyl](methyl)amino}methyl)phenol
1-[7-(1-benzothiophen-3-yl)-9-ethoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methylpropan-1-one
N-[2-(pyridin-3-yloxy)ethyl]-1,3-benzothiazole-6-carboxamide
6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]quinoxaline
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl][2-(2-fluorophenyl)-1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}ethyl]methylamine
2-[2-(1,4-oxazepan-4-ylmethyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
(1S,5R)-6-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2-fluorophenyl)methyl]-3-{2-oxo-2-[4-(thiomorpholin-4-yl)piperidin-1-yl]ethyl}piperazin-2-one
N-benzyl-N-(2-hydroxyethyl)-3-methoxy-4-[(1-methylpiperidin-4-yl)oxy]benzamide
(3S,4R)-4-(4-fluorophenyl)-1-[3-(thiophen-2-yl)propanoyl]pyrrolidine-3-carboxylic acid
(2S,4S)-4-amino-1-(2-amino-4-phenylpyrimidine-5-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
2-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]pyrrolidin-2-yl}ethan-1-ol
N-(1-{1-[2-(cyclohex-1-en-1-yl)acetyl]piperidin-4-yl}-2-phenylethyl)-N-methylpyridine-2-carboxamide
2-amino-N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-4-methyl-1,3-thiazole-5-carboxamide
3-{2-[(3S)-3-hydroxypyrrolidin-1-yl]-2-oxoethyl}-2-methyl-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-4-one
4-(4-{[2-(methoxymethyl)pyrimidin-5-yl]methyl}piperazin-1-yl)-6-methyl-2-(methylsulfanyl)pyrimidine
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
3-(1H-1,3-benzodiazol-1-yl)-1-{4-[4-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}propan-1-one
1-ethyl-N-(2-methoxyethyl)-2-oxo-N-(pyridin-2-ylmethyl)-1,2-dihydropyridine-4-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetamide
2-(furan-2-yl)-1-[1-(2-methoxyphenoxy)propan-2-yl]-1H-imidazole
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-(3-methoxypropyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
(2-methoxyethyl)({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})methylamine
1-[(4aR,8aS)-1-[4-(2-fluorophenyl)benzoyl]-decahydro-1,6-naphthyridin-6-yl]-3-(pyridin-3-yl)propan-1-one
(1S,5R)-6-[(3,5-dimethoxyphenyl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
(2R,3S,6R)-5-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
1-cyclohexyl-N-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide