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1-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-3-(2-oxo-2,3-dihydro-1H-indol-5-yl)urea
N-methyl-4-{3-[(4-methylpiperazin-1-yl)methyl]-1,2,4-oxadiazol-5-yl}aniline
N-(1,3-benzothiazol-6-yl)-4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carboxamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-(pentan-3-yl)-2-(pyridin-3-yl)acetamide
2-[1-(3-methylbut-2-en-1-yl)-4-(quinolin-2-ylmethyl)piperazin-2-yl]ethan-1-ol
N-[(3R,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(2-hydroxyethyl)-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-phenylpyridine-3-carboxamide
N-[(1R)-1-(4-methoxyphenyl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
5-{[benzyl(methyl)amino]methyl}-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)({[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amine
3-(1H-1,3-benzodiazol-1-yl)-1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}propan-1-one
8-(5-methanesulfonyl-2-methylpyrimidin-4-yl)-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N3-[(3,5-difluorophenyl)methyl]-1-(2-methoxyethyl)-4-oxo-N5-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-1-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-yl}ethan-1-one
2-(pyrrolidine-1-carbonyl)-1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine
2-methyl-7-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{[4-(pyrrolidine-1-sulfonyl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
N-[1-(2,5-difluorophenyl)cyclopropyl]-2-ethylpyrimidine-5-carboxamide
(3S,9aR)-3-[(4-methoxyphenyl)methyl]-8-(naphthalene-1-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[2-({3-chloro-6-methylpyrazolo[1,5-a]pyrimidin-2-yl}formamido)ethyl]pyridine-3-carboxamide
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-4-(4-methylphenoxy)piperidine-4-carboxamide
(2S,4R)-4-amino-1-{[5-(cyclohexylsulfanyl)furan-2-yl]methyl}-N-methylpyrrolidine-2-carboxamide
2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-N-[2-(1H-pyrazol-4-yl)ethyl]-2,3-dihydro-1H-isoindole-4-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methyl-1H-pyrazol-1-yl)propan-1-one
2-[1-(1-methanesulfonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]quinolin-4-ol
(2R,3R)-1'-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-3-(1H-imidazol-1-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-[(3R,4S)-1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(1R,2S)-N1-butyl-N2-[2-(1,3-thiazol-4-yl)ethyl]cyclohexane-1,2-dicarboxamide
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(pyrrolidin-1-yl)propan-1-one
2-[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperidin-4-yl]-1,2,3,4-tetrahydroisoquinoline
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-4-phenylbutane-1,2-dione
{4-[(4-methoxyphenyl)methyl]-1-[(4-methylthiophen-2-yl)sulfonyl]piperidin-4-yl}methanol
3-[4-(2,4-dimethylphenyl)piperazine-1-carbonyl]-2-ethyl-1-[(2-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
2-(benzylamino)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
4-[4-(1,3-dimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]-1-methylpiperazin-2-one
2-methyl-1-{4-[4-(3-methylpyridin-2-yl)piperazin-1-yl]piperidin-1-yl}propan-1-one
2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(pyridin-4-ylmethyl)-1,4-dihydropyridine-3-carboxamide
(2S,4R)-4-amino-1-(4-acetamidobenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-1H-indole-5-carboxamide
9-[2-(4-ethoxyphenyl)acetyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]-2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(3aR,6aS)-5-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-fluoro-2-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}quinolin-4-ol
2-methoxy-N-({1-[(2-methyl-1H-imidazol-4-yl)methyl]pyrrolidin-3-yl}methyl)benzamide
3-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-5,5-dimethyl-1,3-oxazolidine-2,4-dione
4-{[(1R,5S,8R)-8-methoxy-3-azabicyclo[3.2.1]octan-3-yl]methyl}-1H-pyrazole-3-carboxylic acid
5-(2,6-dimethylphenoxymethyl)-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
1-[(2-methoxyphenyl)methyl]-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]piperidin-2-one
1-ethyl-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-5-oxopyrrolidine-3-carboxamide