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9-methoxy-7-oxo-3-(2-phenoxypropanoyl)-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
8-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
1-[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
[(8-methoxyquinolin-5-yl)methyl](methyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl]amine
N-(pyridin-4-ylmethyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-amine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-(2-methoxybenzoyl)piperidine
N-[1-(3-methylpyridin-2-yl)propyl]-1H-pyrazole-4-carboxamide
2-[1-(2-methoxyethyl)-3-(2-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-propylpiperidine
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(1H-pyrrole-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
(1S,4S)-2-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptane
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(4-methylpyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-({[4-(dimethylamino)-5-fluoropyrimidin-2-yl]amino}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-({3-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-1H-pyrazol-5-yl}methoxy)phenyl]ethan-1-one
4-{3-[(3-methoxypiperidin-1-yl)methyl]-8-methylimidazo[1,2-a]pyridine-2-carbonyl}morpholine
1-cyclopentyl-6-oxo-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}piperidine-3-carboxamide
2-amino-4-(1-ethyl-1H-indol-4-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(1-{[2-(2,4-dimethoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-pyrazol-4-yl)ethan-1-ol
N-{[5-(pyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
4-methoxy-N-(2-methoxyethyl)-2-{[1-(pyridin-4-ylmethyl)piperidin-4-yl]oxy}benzamide
1'-(quinoxaline-5-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(2-methanesulfonylethyl)amine
2-(2-chlorophenyl)-3-methyl-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-(3-{[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
3-methoxy-N-{1-[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
1-[3-(2H-1,3-benzodioxole-5-carbonyl)piperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}acetamide
5-ethyl-N-(oxolan-2-ylmethyl)-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(1S,5R)-6-{3-methyl-5H,6H-imidazo[2,1-b][1,3]thiazole-2-carbonyl}-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
5-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-N-methyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
(1S,5R)-3-cycloheptanecarbonyl-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-phenyl-1-{[5-(1H-1,2,4-triazole-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidine
N-cyclooctyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-[2-(pyridin-3-yl)ethyl]-9-[3-(1H-1,2,3,4-tetrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N,4-dimethyl-1,3-thiazol-2-amine
8-[(2-chlorophenyl)methyl]-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
1-(ethanesulfonyl)-4-[3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazine
1-[(1-methyl-1H-imidazol-2-yl)methyl]-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
N-[(2-methylphenyl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
N-[(2R,3R)-2-ethoxy-1'-(8-fluoroquinoline-2-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
N-cyclopentyl-2-methyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)propanamide
2-{4-methyl-1-[5-(pyrrolidine-1-carbonyl)furan-2-yl]-1H-1,3-benzodiazol-2-yl}ethan-1-ol
(3S,4R)-1-{[4-(2-aminoethyl)phenyl]methyl}-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
2-(3-hydroxypropyl)-8-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
2,6-difluoro-N-{[7-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
1-methyl-N-{2-[5-methyl-3-(trifluoromethyl)-1H-pyrazol-1-yl]ethyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
2-{2-[1-(pyridin-4-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}acetamide