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N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,4R)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-[({5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-yl}amino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[1-(2,6-dimethylquinoline-4-carbonyl)pyrrolidin-2-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[(2-fluoro-4-methoxyphenyl)methyl]-9-methoxy-N-[(4-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[5-({7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)thiophen-2-yl]prop-2-yn-1-ol
N-[3-(furan-2-yl)phenyl]-1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidine-4-carboxamide
4-ethyl-6-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
(1R,2S)-2-{[5-(2-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}cyclopentan-1-ol
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzamide
1,3-dimethyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1S,6R)-9-[4-(1H-1,2,4-triazol-5-yl)benzoyl]-3,9-diazabicyclo[4.2.1]nonane
2,2-dimethyl-3-{[6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]amino}propan-1-ol
5-(4-methoxy-2-methylphenyl)pyrimidine
N-(1-methyl-1H-indazol-3-yl)-2-[3-(1-methyl-1H-pyrazol-4-yl)-1H-indazol-1-yl]acetamide
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-phenoxypropan-1-one
N-(1H-1,3-benzodiazol-2-yl)-2-[4-(pyrimidin-2-yloxy)piperidin-1-yl]acetamide
2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}quinoline
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-acetamido-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
(2S,4S)-4-amino-1-[2-(5-ethyl-1-benzofuran-3-yl)acetyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-cyclopropyl-1-[(1s,4s)-4-({[4-(2-methylphenyl)phenyl]methyl}amino)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
4-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-propylpyridine
({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)(1-methoxypropan-2-yl)amine
8-(5-hydroxypyridine-2-carbonyl)-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,5S)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-(morpholine-4-carbonyl)piperidine-3-carboxamide
1-{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(thiophene-2-carbonyl)piperidine
4-(3-phenylpropyl)-2-(pyridin-3-yl)morpholine
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(propan-2-yloxy)ethyl]acetamide
ethyl 4-[({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)amino]piperidine-1-carboxylate
5-(2-{2-[(8-chloroquinolin-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-[4-(3-methoxyphenyl)-3-oxopiperazin-1-yl]-2-(thiophen-3-yl)acetic acid
2-[5-({5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}methyl)-2-methoxyphenoxy]acetic acid
3-[1-(pyrazin-2-yl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
1-[1-(2-cyclopropylpyrimidine-5-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
2-(dimethylamino)-8-[(2E)-3-phenylprop-2-en-1-yl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
benzyl(methyl)[1-(pyridin-3-yl)propyl]amine
(4-{[methyl({1H-pyrrolo[2,3-b]pyridin-6-yl})amino]methyl}oxan-4-yl)methanol
(1R,9S)-5-amino-3-(4,5-dimethylfuran-2-yl)-6,12-diazatricyclo[7.2.1.02,7]dodeca-2(7),3,5-triene-4-carbonitrile
3-(2-methoxyethyl)-1-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperidine-3-carboxylic acid
3-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-(propan-2-yl)-1,2-dihydropyridin-2-one
3-{2-[(4-methoxynaphthalen-1-yl)methyl]-5-oxopyrrolidin-2-yl}-N-{2-[2-(trifluoromethyl)phenyl]ethyl}propanamide
4-ethyl-5-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]-1,2,3-thiadiazole
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-1-[2-(piperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methylpyridine-3-carboxamide
1-cyclohexyl-N3-methyl-4-oxo-N5-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-methyl-6-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-(1-ethylpiperidin-4-yl)-N-[1-(pyrazin-2-yl)propan-2-yl]acetamide
3-[(1-acetylpiperidin-4-yl)oxy]-4-methoxy-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]benzamide