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{4-[(2-chlorophenyl)methyl]-1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}methanol
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-(pyrazine-2-carbonyl)pyrrolidin-3-yl]methanol
1-ethyl-4-({5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
1-{1-[(4-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-methoxyphenyl)piperazine
3-{3-[(3-chlorophenyl)methyl]-3-(ethoxycarbonyl)piperidine-1-carbonyl}pyridin-1-ium-1-olate
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
1-[(2-methoxynaphthalen-1-yl)methyl]-4-(prop-2-en-1-yl)-1,4-diazepan-5-one
2-ethyl-9-(2-{methyl[(4-methylphenyl)methyl]amino}acetyl)-2,9-diazaspiro[5.5]undecan-3-one
(3S,4S)-1-[1-(2H-1,3-benzodioxol-5-yl)piperidin-4-yl]-4-(morpholin-4-yl)pyrrolidin-3-ol
2-[1-cyclopentyl-3-(2-methylphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
1-[4-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
(1S,3R)-3-amino-N-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}cyclopentane-1-carboxamide
2-[4-(1-benzothiophen-3-yl)-2-(morpholin-4-ylmethyl)phenoxy]-N-[1-(thiophen-2-yl)ethyl]acetamide
1-(2-fluorophenyl)-4-[(2S,4S)-4-[(4-fluorophenyl)sulfanyl]-1-(1-methylpiperidin-4-yl)pyrrolidine-2-carbonyl]piperazine
(2S)-2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-methylbutanamide
N-[2-(3-methoxyphenyl)-1-[1-(thiophene-3-carbonyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
8-(furan-3-ylmethyl)-1-(3-methylbutyl)-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[6-(4-methylpiperazin-1-yl)pyridine-3-carbonyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-{[8-(1-benzofuran-2-carbonyl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}-2-fluorobenzamide
2,3-dimethyl-N-[(1-propyl-1H-imidazol-2-yl)methyl]quinoxaline-6-carboxamide
1-[6-hydroxy-4-(1H-imidazol-4-ylmethyl)-1,4-diazepan-1-yl]-2-[methyl(propan-2-yl)amino]ethan-1-one
N-methyl-2-[2-oxo-3-(trifluoromethyl)-1,2-dihydropyridin-1-yl]-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)acetamide
1-[2-(5-methyl-4-{[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-1-yl)ethyl]piperidine
2-{4-[2-(dimethylamino)phenyl]-1H-pyrazol-1-yl}propanamide
(3S,5R)-1-benzyl-5-(4-methylpiperazine-1-carbonyl)piperidine-3-carboxylic acid
(2R,4S)-1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}-4-hydroxypiperidine-2-carboxylic acid
({[7-(3,5-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}sulfamoyl)dimethylamine
3-ethyl-1-(1H-indazol-5-yl)-3-(2,2,2-trifluoroethyl)urea
N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
4-(2-methoxybutanoyl)-1-(3-methoxyphenyl)piperazin-2-one
(1S,5R)-6-(3-fluoro-4-methylbenzoyl)-3-methyl-3,6-diazabicyclo[3.2.2]nonane
(2,1,3-benzothiadiazol-5-ylmethyl)({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
(2R)-N-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}oxolane-2-carboxamide
N-benzyl-2-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-sulfonamide
2,2-dimethyl-N-(1-{1-[2-(morpholin-4-yl)ethyl]piperidin-4-yl}-1H-pyrazol-5-yl)propanamide
2-[4-(2,5-dioxo-4-propylimidazolidin-4-yl)piperidin-1-yl]acetic acid
3-cyclobutyl-5-{[5-(oxan-2-yl)furan-2-yl]methyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[(3,4-dimethoxyphenyl)methyl]-N-(1,4-dioxan-2-ylmethyl)-1,3-benzoxazole-6-carboxamide
1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-3-(1,3-dimethyl-1H-pyrazol-5-yl)urea
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1R,2S)-2-(methoxymethyl)cyclopentyl]propanamide
[1-(adamantan-1-yl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-(pyridin-3-ylmethyl)-1,4-diazepane
5-chloro-2-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]phenol
1-cyclopentyl-4-oxo-N3-(prop-2-en-1-yl)-N5-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[3-(4-fluorophenoxy)propyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
ethyl 1-[(3-chloro-4-methoxyphenyl)carbamoyl]-4-(2-phenylethyl)piperidine-4-carboxylate
methyl 1-(2-methoxyethyl)-5-[(4-methylpentan-2-yl)amino]-3-(3-phenylpropanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}amine
N-benzyl-3-[(3,4-dimethylpiperazin-1-yl)methyl]-N-methylimidazo[1,2-a]pyridine-2-carboxamide