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1-benzyl-4-oxo-N3-[(1-phenylcyclopentyl)methyl]-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-[3-(1H-pyrazol-1-yl)propyl]piperidine-2-carboxamide
1-methyl-1'-[2-(methylamino)-1,3-thiazole-4-carbonyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-(2-phenylpropyl)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine
N-{1-[1-(cyclobutylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methoxybenzamide
7-methyl-2-(2-phenoxyethanesulfonyl)-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-6-(4-methylpyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-({7-[(2,3-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2-methylbutanamide
4'-[(5-chloro-2-fluorophenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-{[1-(2-methoxyethyl)-1H-imidazol-2-yl]methyl}-2-(1,3-thiazol-2-yl)piperidine
8-(3-methylpentanoyl)-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(4-fluorophenyl)-4-{[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methyl}piperazine
methyl 3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-[(4-fluorophenyl)methoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(2-methylphenyl)acetamide
2-{4-[2-(8-chloro-2-ethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetyl]piperazin-1-yl}-N,N-dimethylacetamide
N-methyl-6-oxo-4-[4-(1H-1,2,4-triazol-1-yl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
2-(4-cyclopentyl-1,4-diazepan-1-yl)-2-[4-(1H-pyrazol-1-yl)phenyl]acetic acid
methyl 3-acetamido-5-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
8-(3-hydroxybenzoyl)-3-(3-methylbutyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2-chlorophenyl)-4-[2-(2-ethoxyphenyl)acetyl]piperazin-2-one
1-methyl-4-{1-[1-(1,3-thiazol-2-yl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
N-[4-(furan-2-yl)phenyl]-1-(2-oxo-2-phenylacetyl)piperidine-3-carboxamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-3-{2-[(2-fluoro-4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
(4aS,7aR)-1-(1-ethyl-1H-pyrazole-4-carbonyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4S)-3-{2-[3-(benzyloxy)azetidin-1-yl]-2-oxoethyl}-4-phenyl-1,3-oxazolidin-2-one
N-cyclopropyl-4-methoxy-2-{[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]oxy}benzamide
4-[2-(cyclopentylmethyl)-3H-imidazo[4,5-b]pyridin-3-yl]-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidine
N,N-diethyl-1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazole-5-carboxamide
4-methyl-2-{1-[4-(methylsulfanyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1H-imidazole
4-(furan-3-ylmethyl)-3-[2-oxo-2-(4-phenylpiperazin-1-yl)ethyl]piperazin-2-one
5-[(4-fluorophenyl)methyl]-5-{1-[2-(3-methylphenyl)acetyl]piperidin-4-yl}-3-(oxolan-3-yl)imidazolidine-2,4-dione
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-ethyl-2-oxo-N-{2-[(trifluoromethyl)sulfanyl]ethyl}-1,2-dihydropyridine-4-carboxamide
6-[(3-methoxyphenyl)methoxy]-1-(2-methylpropyl)-4-[2-(pyridin-3-yl)acetyl]-1,4-diazepan-2-one
N-benzyl-5-({methyl[1-(pyridin-2-yl)ethyl]amino}methyl)pyrimidin-2-amine
2-(4-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[(2-methylphenyl)methyl]piperazin-2-yl)ethan-1-ol
1-(6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridin-3-yl)ethan-1-one
ethyl 5-({[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-pyrazole-4-carboxylate
2-[4-(2-ethylpyrimidine-5-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
dimethyl(3-{2-[1-(morpholine-2-carbonyl)piperidin-4-yl]-1H-imidazol-1-yl}propyl)amine
3,5-dichloro-4-[1-(oxan-2-ylmethyl)-1H-imidazol-2-yl]pyridine
3-{2-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
N-cyclohexyl-1,3-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1S,5R)-6-[6-(methoxymethyl)pyridine-2-carbonyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
N4-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N4,5-dimethylpyrimidine-2,4-diamine
1-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-ethylurea
N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
4-methyl-N-{[1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-[1-cyclopentyl-3-(4-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methyl]acetamide
N-[(4-fluorophenyl)methyl]-3-{1-[2-(thiophen-3-yl)acetyl]piperidin-4-yl}propanamide