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2-[(5-methyl-1H-1,3-benzodiazol-2-yl)sulfanyl]-N-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}acetamide
[(3R,4R)-1-(2-methoxypyridine-3-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
4-hydroxy-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
3-[1-(5-methoxyfuran-2-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
1-benzyl-8-[(4-hydroxy-3,5-dimethoxyphenyl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-1,2,3,4-tetrahydroisoquinoline
5-[(3-ethyl-1H-1,2,4-triazol-1-yl)methyl]-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
(1S,4R)-2-[3-(4-fluorophenoxy)propyl]-2-azabicyclo[2.2.1]heptan-3-one
N-[5-({3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}sulfonyl)-1,3-thiazol-2-yl]acetamide
methyl 4-{4-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]piperazin-1-yl}benzoate
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(2-oxopyrrolidin-1-yl)benzamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(2-methoxy-6-methylbenzoyl)pyrrolidin-3-yl]methanol
4-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)benzene-1-sulfonamide
[(2-methyl-1,3-thiazol-4-yl)methyl](1-phenoxypropan-2-yl)amine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
1-[(2-chloro-6-fluorophenyl)methyl]-5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-methyl-1H-1,2,4-triazole
N-[1-(cyclohexylmethyl)piperidin-3-yl]-2-(dimethylamino)acetamide
methyl 3-(furan-3-amido)-6-[(3-phenylpiperidin-1-yl)methyl]thieno[2,3-b]pyridine-2-carboxylate
4-(3-chlorophenoxy)-1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
8-methyl-2-({3-oxo-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-4-yl}methyl)-4H-pyrido[1,2-a]pyrimidin-4-one
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(thiophen-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
3-(1-methyl-1H-imidazol-2-yl)-6-[3-(3-methylphenoxymethyl)piperidin-1-yl]pyridazine
2-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-4-methylphenol
(2E)-N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-3-(4-methoxyphenyl)-N-methylprop-2-enamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2H-1,3-benzodioxole-5-carboxamide
1-[1,3-dioxo-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]piperidine-4-carboxamide
N-benzyl-3-cyano-N-(3-hydroxy-2-methylpropyl)benzamide
3-phenyl-7-[(2,4,5-trimethylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
N-(1-{4-[methyl({[2-(trifluoromethyl)phenyl]methyl})carbamoyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]isoquinoline-1-carboxamide
2-(3-aminopropanoyl)-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,4-dihydro-2H-1-benzopyran-3-carboxamide
{4-[5-(4-phenylazepane-1-carbonyl)pyridin-2-yl]phenyl}methanol
N-[3-({[(2,4-dimethoxy-3-methylphenyl)methyl]amino}methyl)-5-(pyrrolidine-1-carbonyl)phenyl]acetamide
N-(1H-imidazol-2-ylmethyl)-N,6-dimethyl-2-(pyridin-3-yl)pyrimidin-4-amine
4,6,7-trimethyl-2-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]quinazoline
[1-({4-[(2E)-2-methylbut-2-en-1-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidin-2-yl]methanol
3-(1-benzyl-1H-pyrazol-4-yl)-2-methoxypyridine
N-[(2-methoxyphenyl)methyl]-2-{[(1R,2S)-2-phenylcyclopropyl]amino}acetamide
1-[2-(dimethylamino)ethyl]-4-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
ethyl 2-[methyl({[1-(oxolan-2-ylmethyl)-2-(propane-1-sulfonyl)-1H-imidazol-5-yl]methyl})amino]acetate
(2S,4S,5R)-4-[(2-methoxyethyl)carbamoyl]-1,2-dimethyl-5-(2-methylphenyl)pyrrolidine-2-carboxylic acid
1-(4-acetylphenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
5-[1-(2,5-difluorobenzoyl)piperidin-4-yl]-5-[(3-fluorophenyl)methyl]-3-(2-methoxyethyl)imidazolidine-2,4-dione
2-(3-{[cyclohexyl(ethyl)amino]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
3-(2-oxo-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)-1,3-thiazolidine-2,4-dione
2-[(5-benzyl-4-phenyl-1H-imidazol-1-yl)methyl]pyridine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}({[1-(prop-2-en-1-yl)pyrrolidin-3-yl]methyl})amine