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N-[(4-fluoro-3-methoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
7-(2-methoxyethyl)-2-(1,2-thiazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-4-{3-[4-(pyridin-4-yloxy)piperidine-1-carbonyl]phenyl}butan-2-ol
3-(2-methoxybenzoyl)-1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
N,6-dimethyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydroquinoline-4-carboxamide
2-{1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-3-carbonyl}pyridine
N-[(3R,4R)-1-(1-benzofuran-2-ylmethyl)-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
2-[(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperidin-3-yl)methyl]-1H-1,3-benzodiazole
4-(3-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}propanamido)benzamide
1-[(2-butyl-1H-imidazol-4-yl)methyl]-3-[3-(trifluoromethyl)benzoyl]piperidine
N-[(3S,5S)-5-(ethylcarbamoyl)-1-[(3-fluorophenyl)methyl]pyrrolidin-3-yl]pyrazine-2-carboxamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-cyclopropyl-N-[2-(diethylamino)ethyl]-N-ethyl-1H-pyrazole-4-carboxamide
[(4-chlorophenyl)methyl][(8-methyl-2-{octahydropyrrolo[1,2-a]piperazin-2-yl}quinolin-3-yl)methyl]amine
N-[1-(3-phenylpropyl)piperidin-3-yl]quinoxaline-6-carboxamide
methyl 5-{[(2,4-difluorophenyl)methyl]amino}-3-acetamido-1-methyl-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{2-[2-(3-chloro-2,6-difluorophenyl)-1H-imidazol-1-yl]ethyl}-5-cyclopropyl-1,2,4-oxadiazole
(2S,4S)-4-amino-1-[(6-chloropyridin-3-yl)methyl]-N,N-diethylpyrrolidine-2-carboxamide
{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}(methyl)[2-(pyridin-4-yl)ethyl]amine
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}urea
[(2S,6S)-11-methoxy-4-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
N-methyl-5-{[4-(piperidin-1-yl)butanamido]methyl}-1,2,4-oxadiazole-3-carboxamide
1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3-(methanesulfonylmethyl)piperidine
{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
4-(2-methoxyphenoxy)-1-(5-propylpyrimidin-4-yl)piperidine-4-carboxylic acid
6-amino-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]pyridine-3-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-4H-thieno[3,2-b]pyrrole-5-carboxamide
3-(1,3-benzoxazol-2-yl)-N-benzylpiperidine-1-sulfonamide
1-[(2,3-difluorophenyl)methyl]-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-1H-pyrazole-4-carboxamide
3-[(3R,4S)-1-(4-fluoro-2-methylbenzoyl)-4-(morpholin-4-yl)piperidin-3-yl]propan-1-ol
2-(3-chlorophenyl)-1-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
3-(1-{imidazo[1,2-a]pyridine-6-carbonyl}piperidin-4-yl)-1,3-oxazolidin-2-one
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(3-methyl-1H-pyrazole-5-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[2-(2-methoxyethyl)pyrimidin-5-yl]methyl}-N-methyl-1-(3-phenylpropyl)piperidin-3-amine
N-cyclopropyl-N-[(3-hydroxyphenyl)methyl]-2,6-dimethylpyridine-4-carboxamide
2-{[4-(3-methoxyphenyl)-5-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
3-{2-[4-(4-fluorophenyl)piperazin-1-yl]-2-oxoethyl}-1-methyl-3-(4-phenylphenyl)pyrrolidine-2,5-dione
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
(1R,5R)-3-(1-phenylcyclopropanecarbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
7-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-N,N-dimethyl-2-phenylacetamide
2-[1-(3-methylbutyl)-4-{[4-(trifluoromethyl)phenyl]methyl}piperazin-2-yl]ethan-1-ol
(3aS,6aS)-2-cyclopentanecarbonyl-5-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-{[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl](propan-2-yl)amino}-2-(4-methoxy-3,5-dimethylphenyl)acetic acid
5-(2-methoxy-4-methylphenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-hydroxy-N-{1-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(3-methylphenyl)pyrimidine-5-carboxamide
ethyl 4-{[4-(3-cyclohexylpropanoyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-2-(4-propanoylphenoxy)acetamide
N-cyclohexyl-N-(2-hydroxy-2-phenylethyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
4-{[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]methyl}-2-(propan-2-yl)pyrimidine