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4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]-1-[(2-methylphenyl)methyl]piperidine
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3,5-dimethyl-1H-pyrazol-1-yl)propanamide
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2-methyl-4-phenylpyrimidine
ethyl 1-[7-cyclobutaneamido-1-methyl-2-(pyridin-4-yl)-1H-1,3-benzodiazole-5-carbonyl]piperidine-4-carboxylate
2-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-[4-(propan-2-yl)morpholin-2-yl]ethan-1-one
2-methyl-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-5-(propan-2-yl)furan-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(3-chloro-1,2-oxazol-5-yl)propanamide
5-{1-[3-(dimethylamino)benzoyl]piperidin-4-yl}-3-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-propylimidazolidine-2,4-dione
1-amino-N-[1-(4-methoxyphenyl)propyl]cyclopropane-1-carboxamide
3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
3-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]azetidin-3-yl}pyridine
3-{4-[1-(methoxymethyl)cyclobutanecarbonyl]piperazin-1-yl}-2,5-dimethylpyrazine
N-methyl-N-[(3-methylpyridin-2-yl)methyl]-2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)butanamide
2-cyclopropanecarbonyl-8-(2-ethylbenzoyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
5-(3-ethyl-1,2,4-oxadiazol-5-yl)-1-[(3-fluorophenyl)methyl]piperidin-2-one
methyl 2-(1-{[2-(4-fluorophenoxy)pyridin-3-yl]carbamoyl}pyrrolidin-3-yl)acetate
1-(3-chloro-4-fluorophenyl)-3-(2-methoxyethyl)-5-[2-(oxolan-2-yl)ethyl]-1H-1,2,4-triazole
N-(2,3-dihydro-1H-inden-2-yl)-N-methyl-2-(morpholin-4-yl)pyrimidine-5-carboxamide
(2E)-N-{[7-(6-methoxypyridazin-3-yl)-5-methyl-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(pyridin-4-yl)prop-2-enamide
2-[2,5-dioxo-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidin-3-yl]-N-methyl-N-(2-phenylethyl)acetamide
N-{4-[cyclopropyl(pyridin-4-ylmethyl)carbamoyl]phenyl}-2-methylfuran-3-carboxamide
5-(4-methoxyphenyl)-N-{1-[2-(methylsulfanyl)ethyl]piperidin-4-yl}furan-2-carboxamide
N-[1-(furan-2-carbonyl)piperidin-3-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(3R,4S)-1-(2-methanesulfonylethyl)-N,N-dimethyl-4-(5-methylfuran-2-yl)pyrrolidin-3-amine
1-methyl-3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}-3-(4-phenylphenyl)pyrrolidine-2,5-dione
2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(5-methylthiophen-2-yl)methyl]acetamide
(2-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}phenyl)methanol
5-(4-methoxyphenyl)-N-{[1-(2-phenylethyl)piperidin-4-yl]methyl}-1,2,4-triazin-3-amine
N-methyl-1-(propan-2-yl)-N-(quinoxalin-6-ylmethyl)-1H-pyrazole-4-carboxamide
(9aS)-N-[2-(propan-2-yl)phenyl]-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carboxamide
2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}-N-(pyridin-2-ylmethyl)acetamide
2-[6-oxo-4-(piperazin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[3-(oxolan-3-yl)propyl]acetamide
methyl (2S,4S)-1-[(2,5-difluorophenyl)methyl]-4-[2-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
2-{4-[1-(butan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenoxy}-1-(morpholin-4-yl)ethan-1-one
3-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
2-(1-methyl-1H-indol-3-yl)-N-[(3-methyl-5-oxo-4,5-dihydro-1H-pyrazol-4-yl)methyl]acetamide
2-(2-methoxyethyl)-8-[4-(trifluoromethyl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(1-methanesulfonylpiperidin-3-yl)methyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
N-[(2-ethoxyphenyl)methyl]-2-methyl-N-(prop-2-en-1-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
4-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
methyl 2-{N-methyl-1-[2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazol-4-yl]formamido}acetate
methyl 4-(5-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1-methyl-1,2-dihydroquinolin-2-one
3-[(3R,4S)-1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-ethyl-2-[3-(4-phenylbenzoyl)piperidin-1-yl]acetamide
1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidine
N-{1-[1-(5-ethyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
1-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine