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N,3,5-trimethyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-4-carboxamide
N-({8-[(3-ethoxy-2-hydroxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)oxolane-2-carboxamide
(2R,6R)-4-(dimethyl-1,2-oxazole-4-carbonyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-(4-benzyl-2-oxopyrrolidin-1-yl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylacetamide
3-methoxy-1-{2-oxo-2-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl]ethyl}-1,2-dihydropyridin-2-one
2-(2-aminoethyl)-N-{[3-(4-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
ethyl 1-benzyl-5-(2-methylfuran-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
N-(2,5-dimethylphenyl)-3-{[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}propanamide
2-(4-fluorophenyl)-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
6-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]pyridine-2-carboxylic acid
2-methyl-1-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]propan-1-one
4-[4-(2-fluorophenoxy)piperidin-1-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-2-amine
1-[(2R)-oxolan-2-ylmethyl]-4-(5-propylfuran-2-yl)-1H-1,2,3-triazole
1-benzyl-N-[2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
(3R,4R)-1-(2,6-dimethylpyridin-4-yl)-3,4-dimethylpyrrolidin-3-ol
1-(5-methyl-1,3-oxazole-4-carbonyl)-4-[(methylsulfanyl)methyl]piperidine
5-[1-(3,4-dimethoxybenzoyl)piperidin-4-yl]-3-(oxolan-2-ylmethyl)-5-propylimidazolidine-2,4-dione
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[2-(thiophen-2-yl)ethyl]piperidine
4-(2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetyl)-1,4-diazepane-1-carbaldehyde
1-ethyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}piperidine-3-carboxamide
1-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazole-3-carbonyl]-2-(pyrrolidine-1-carbonyl)piperazine
3-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidine-1-carbonyl]pyridin-2-ol
2-(1,3-benzoxazol-2-yl)-N-[2-(furan-2-yl)ethyl]acetamide
N-methyl-N-[3-(morpholin-4-yl)propyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-hydroxy-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-1,2-oxazole-5-carboxamide
5-[(4-fluorophenyl)methyl]-5-{1-[(4-hydroxyphenyl)methyl]piperidin-4-yl}-3-(2-methoxyethyl)imidazolidine-2,4-dione
3-(2-fluoro-4-methoxyphenyl)-1-methyl-1-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
2-butoxy-1-{2,7-diazaspiro[4.5]decan-7-yl}ethan-1-one
N-(4-fluoro-2-methylphenyl)-3-(1-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)propanamide
2-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-[1-(4-fluorophenyl)piperidin-4-yl]acetamide
5-{[2-(adamantan-1-yl)ethyl](methyl)amino}-1-[(3,4-difluorophenyl)methyl]azepan-2-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperidin-3-amine
(4-{5-[1-(propan-2-yloxy)ethyl]-1,2,4-oxadiazol-3-yl}phenyl)methanol
2-[(5-methylpyrazin-2-yl)methyl]-9-(3-methylthiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)but-3-enamide
5-[(2-fluoro-5-methoxyphenyl)methyl]-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
3-[(3R,4S)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(3S,4S)-4-(4-fluorophenyl)-1-{[2-(2-hydroxyethoxy)phenyl]methyl}piperidin-3-ol
N-(3-chloro-4-methoxyphenyl)-3-{1-[(4-methoxyphenyl)methyl]piperidin-3-yl}propanamide
2-methyl-2-(2-{methyl[(1-methylpyrrolidin-3-yl)methyl]amino}-4-(morpholin-4-yl)pyrimidin-5-yl)propanoic acid
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide
N-[(2-{4-[5-(methoxymethyl)furan-2-amido]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N-{1-[(3,5-difluorophenyl)methyl]piperidin-4-yl}-3-(pyridin-4-yl)propanamide
N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(methoxymethyl)thiophene-2-carboxamide
4-methyl-6-{6-[(pyridin-2-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidin-2-amine
3-(8-methoxy-2-methylquinolin-5-yl)-1-methyl-6-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N,N-bis(1,3-oxazol-4-ylmethyl)-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
5-fluoro-8-[4-(morpholine-4-carbonyl)pyridin-2-yl]quinoline