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N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-3-(pyridin-4-yl)propanamide
3-cyclopropyl-5-({[(2-methylphenyl)methyl]sulfanyl}methyl)-1H-1,2,4-triazole
2-{[3-(pyridin-3-yl)azetidin-1-yl]methyl}benzonitrile
N-[2-(furan-2-yl)ethyl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidin-2-amine
1-(4-{[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenyl)ethan-1-one
N-[1-(dimethylsulfamoyl)azepan-3-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
3-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}phenol
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-4-(4-methoxyphenyl)butane-1,4-dione
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(1-propylpiperidin-4-yl)piperidine
N-({3-[(4-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
1-[(2S)-oxolane-2-carbonyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
N3-[(2-fluorophenyl)methyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
methyl 3-{[(5-ethyl-1,2-oxazol-3-yl)formamido]methyl}-5-(4-fluorobenzamido)benzoate
methyl 3-[(2-fluorophenyl)methyl]-7-oxo-9-(thiophen-3-ylmethoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
3-(2,5-dimethylphenyl)-4-(1H-imidazol-2-yl)-1H-pyrazole
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cycloheptanecarboxamide
3-[(3R,4S)-1-[(3-fluorophenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
1-[3-(hydroxymethyl)-3-(2-methoxyethyl)piperidin-1-yl]-3-methanesulfonylpropan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-1-[4-(3-methylphenoxy)piperidin-1-yl]propan-1-one
(1S,5R)-6-(cyclobutylmethyl)-3-(5-methylpyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,7S)-N-methyl-3-[(3-methylphenyl)methyl]-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-{1-[(5-ethylpyridin-2-yl)methyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-[1-(thiophen-3-yl)propan-2-yl]piperidin-4-amine
N-{[7-(4-methyl-2-oxopentanoyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}pyridine-4-carboxamide
N-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}-2-(thiophene-2-sulfonamido)acetamide
1-benzyl-N3-methyl-4-oxo-N3-(2-phenylethyl)-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[2-(morpholin-4-yl)-2-(pyridin-2-yl)ethyl]acetamide
N-[(1-cyclopropanecarbonylpiperidin-4-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-{3-[(2,6-dimethylphenyl)carbamoyl]phenyl}-4-methylpyridine-3-carboxamide
N-cyclopropyl-5-{1-[3-(1H-pyrrol-1-yl)propanoyl]pyrrolidin-2-yl}thiophene-2-carboxamide
(2R,3R,6R)-5-(5-ethyl-2-methylpyrimidin-4-yl)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-(2,3-dihydro-1-benzofuran-5-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S,4R)-1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-methylthiophen-2-yl)piperidin-3-ol
5-[5-(3-methylphenyl)furan-2-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
1-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenylpiperidine
2-{1-butyl-5-[(3-oxo-2,3-dihydro-1H-isoindol-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidine
(1R,5R)-6-[(3,4-difluorophenyl)methyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
1-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-4-(pyrrolidin-1-yl)pentan-1-one
5-(1-{[5-chloro-1-methyl-3-(5-methyl-1,2-oxazol-3-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
8-(4,6-dimethylpyridine-3-carbonyl)-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-4-{4-[(N-methyl-1-thiophen-2-ylformamido)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
3-(2H-1,3-benzodioxol-5-yl)-3-phenyl-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}propanamide
1-[2-({2-methylthieno[3,2-d]pyrimidin-4-yl}amino)ethyl]imidazolidin-2-one
4-cyclobutyl-11-methyl-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)quinolin-4-ol
2,4-dimethoxy-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-ethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-[(2-methylpropyl)amino]pyridine-3-carboxamide